TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataKi: 8.30E+3nMAssay Description:Competitive inhibition of recombinant human MAO-B using farnesylamine as substrate by horseradish peroxidase-Amplex red-coupled assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 189nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 550nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 650nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 1.39E+3nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 1.87E+3nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 1.97E+3nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 3.39E+3nMAssay Description:The compound was tested for its inhibitory activity against platelet aggregationMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 3.87E+3nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 4.33E+3nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 4.57E+3nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 5.38E+3nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 5.52E+3nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 5.87E+3nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 6.21E+3nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 6.24E+3nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 6.91E+3nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 6.91E+3nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 7.22E+3nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 9.33E+3nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 9.55E+3nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 1.41E+4nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 1.54E+4nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 3.14E+4nMAssay Description:Antagonistic activity against VLA-4 binding to recombinant human VCAM by ramos cell assayMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 4.27E+4nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Hefei University of Technology
Curated by ChEMBL
Hefei University of Technology
Curated by ChEMBL
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured over 15 mins by ...More data for this Ligand-Target Pair