TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 6.5nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C zeta type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-zeta expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-epsilon expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate a...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 71nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-epsilon expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate a...More data for this Ligand-Target Pair
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-epsilon expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate a...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-epsilon expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate a...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-epsilon expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate a...More data for this Ligand-Target Pair
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-epsilon expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate a...More data for this Ligand-Target Pair
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-epsilon expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate a...More data for this Ligand-Target Pair
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-epsilon expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate a...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-epsilon expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate a...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-alpha expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate aft...More data for this Ligand-Target Pair
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-epsilon expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate a...More data for this Ligand-Target Pair
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-epsilon expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate a...More data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-epsilon expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate a...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-epsilon expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate a...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetProtein kinase C iota type(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of full-length N-terminal GST-fused human PKC-iota expressed in baculovirus expression system using (5FAM) RFARKGSLRQKNV as substrate afte...More data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Agency for Science, Technology and Research (A*STAR)
Curated by ChEMBL
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair