Compile Data Set for Download or QSAR
Found 13 Enz. Inhib. hit(s) with all data for entry = 50002811
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Nanjing University of Technology

Curated by ChEMBL
LigandPNGBDBM50143558(CHEMBL41355 | EZOGABINE | N-(2-amino-4-(4-fluorobe...)copy SMILEScopy InChI
Affinity DataEC50:  350nMAssay Description:Channel opening activity at KCNQ2 (unknown origin) expressed in CHO cells after 10 mins by atomic absorption spectrophotometry-based Rb+ flow assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Nanjing University of Technology

Curated by ChEMBL
LigandPNGBDBM50463338(CHEMBL4244768)copy SMILEScopy InChI
Affinity DataEC50:  300nMAssay Description:Channel opening activity at KCNQ2 (unknown origin) expressed in CHO cells after 10 mins by atomic absorption spectrophotometry-based Rb+ flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H997WBPubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Nanjing University of Technology

Curated by ChEMBL
LigandPNGBDBM50463339(CHEMBL4250839)copy SMILEScopy InChI
Affinity DataEC50:  140nMAssay Description:Channel opening activity at KCNQ2 (unknown origin) expressed in CHO cells after 10 mins by atomic absorption spectrophotometry-based Rb+ flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H997WBPubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Nanjing University of Technology

Curated by ChEMBL
LigandPNGBDBM50463340(CHEMBL4244025)copy SMILEScopy InChI
Affinity DataEC50:  2.93E+3nMAssay Description:Channel opening activity at KCNQ2 (unknown origin) expressed in CHO cells after 10 mins by atomic absorption spectrophotometry-based Rb+ flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H997WBPubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Nanjing University of Technology

Curated by ChEMBL
LigandPNGBDBM50463341(CHEMBL4238783)copy SMILEScopy InChI
Affinity DataEC50:  20nMAssay Description:Channel opening activity at KCNQ2 (unknown origin) expressed in CHO cells after 10 mins by atomic absorption spectrophotometry-based Rb+ flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H997WBPubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Nanjing University of Technology

Curated by ChEMBL
LigandPNGBDBM50463342(CHEMBL4247002)copy SMILEScopy InChI
Affinity DataEC50:  40nMAssay Description:Channel opening activity at KCNQ2 (unknown origin) expressed in CHO cells after 10 mins by atomic absorption spectrophotometry-based Rb+ flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H997WBPubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Nanjing University of Technology

Curated by ChEMBL
LigandPNGBDBM50463349(CHEMBL4250878)copy SMILEScopy InChI
Affinity DataEC50:  20nMAssay Description:Channel opening activity at KCNQ2 (unknown origin) expressed in CHO cells after 10 mins by atomic absorption spectrophotometry-based Rb+ flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H997WBPubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Nanjing University of Technology

Curated by ChEMBL
LigandPNGBDBM50463344(CHEMBL4246564)copy SMILEScopy InChI
Affinity DataEC50:  250nMAssay Description:Channel opening activity at KCNQ2 (unknown origin) expressed in CHO cells after 10 mins by atomic absorption spectrophotometry-based Rb+ flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H997WBPubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Nanjing University of Technology

Curated by ChEMBL
LigandPNGBDBM50463345(CHEMBL4247074)copy SMILEScopy InChI
Affinity DataEC50:  34nMAssay Description:Channel opening activity at KCNQ2 (unknown origin) expressed in CHO cells after 10 mins by atomic absorption spectrophotometry-based Rb+ flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H997WBPubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Nanjing University of Technology

Curated by ChEMBL
LigandPNGBDBM50463346(CHEMBL4250403)copy SMILEScopy InChI
Affinity DataEC50:  30nMAssay Description:Channel opening activity at KCNQ2 (unknown origin) expressed in CHO cells after 10 mins by atomic absorption spectrophotometry-based Rb+ flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H997WBPubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Nanjing University of Technology

Curated by ChEMBL
LigandPNGBDBM50463347(CHEMBL4246596)copy SMILEScopy InChI
Affinity DataEC50:  120nMAssay Description:Channel opening activity at KCNQ2 (unknown origin) expressed in CHO cells after 10 mins by atomic absorption spectrophotometry-based Rb+ flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H997WBPubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Nanjing University of Technology

Curated by ChEMBL
LigandPNGBDBM50463348(CHEMBL4246239)copy SMILEScopy InChI
Affinity DataEC50:  290nMAssay Description:Channel opening activity at KCNQ2 (unknown origin) expressed in CHO cells after 10 mins by atomic absorption spectrophotometry-based Rb+ flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H997WBPubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Nanjing University of Technology

Curated by ChEMBL
LigandPNGBDBM50463343(CHEMBL4242757)copy SMILEScopy InChI
Affinity DataEC50:  1.08E+3nMAssay Description:Channel opening activity at KCNQ2 (unknown origin) expressed in CHO cells after 10 mins by atomic absorption spectrophotometry-based Rb+ flow assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H997WBPubMed