Compile Data Set for Download or QSAR
Found 135 Enz. Inhib. hit(s) with all data for entry = 50002886
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464412(CHEMBL4278248)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464415(CHEMBL4278575)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464412(CHEMBL4278248)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50035179(Agomelatine | CHEMBL10878 | N-[2-(7-Methoxy-naphth...)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464406(CHEMBL4280601)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464420(CHEMBL4290302)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464407(CHEMBL4292336)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464402(CHEMBL4279639)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464411(CHEMBL4291381)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464409(CHEMBL4283539)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464402(CHEMBL4279639)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464403(CHEMBL4294790)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464417(CHEMBL4280791)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464400(CHEMBL4293386)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464414(CHEMBL4288497)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50035179(Agomelatine | CHEMBL10878 | N-[2-(7-Methoxy-naphth...)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMedDrugBank
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464413(CHEMBL4281712)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464400(CHEMBL4293386)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464405(CHEMBL4281915)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464415(CHEMBL4278575)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464405(CHEMBL4281915)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464418(CHEMBL4284223)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464421(CHEMBL4286896)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464399(CHEMBL4278446)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464404(CHEMBL4286494)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464416(CHEMBL4289115)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464408(CHEMBL4285145)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464413(CHEMBL4281712)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464402(CHEMBL4279639)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464414(CHEMBL4288497)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464407(CHEMBL4292336)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464402(CHEMBL4279639)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464421(CHEMBL4286896)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464419(CHEMBL4277185)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464406(CHEMBL4280601)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464409(CHEMBL4283539)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464417(CHEMBL4280791)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464411(CHEMBL4291381)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464423(CHEMBL4288925)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464408(CHEMBL4285145)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464420(CHEMBL4290302)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464422(CHEMBL4277390)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464401(CHEMBL4288690)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464410(CHEMBL4292109)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464423(CHEMBL4288925)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464405(CHEMBL4281915)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464410(CHEMBL4292109)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464405(CHEMBL4281915)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464419(CHEMBL4277185)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464403(CHEMBL4294790)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
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