Compile Data Set for Download or QSAR
Found 46 Enz. Inhib. hit(s) with all data for entry = 50002930
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)copy SMILEScopy InChI
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor (unknown origin) in cerebral cortex membranes after 60 mins by TopCount scintillation counting ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMedDrugBank
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464861(CHEMBL4291322)copy SMILEScopy InChI
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]LSD from recombinant human 5-HT7 receptor expressed in CHO cell membranes after 120 mins by TopCount scintillation counting metho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50150105(CHEMBL124069 | [2-(6-Fluoro-chroman-8-yloxy)-ethyl...)copy SMILEScopy InChI
Affinity DataKi:  0.470nMAssay Description:Inhibition of serotonin reuptake in SERT (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464861(CHEMBL4291322)copy SMILEScopy InChI
Affinity DataKi:  0.530nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HEK293 cell membranes after 60 mins by TopCount scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464857(CHEMBL4277476)copy SMILEScopy InChI
Affinity DataKi:  0.550nMAssay Description:Displacement of [3H]LSD from recombinant human 5-HT7 receptor expressed in CHO cell membranes after 120 mins by TopCount scintillation counting metho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464863(CHEMBL4285796)copy SMILEScopy InChI
Affinity DataKi:  0.790nMAssay Description:Displacement of [3H]LSD from recombinant human 5-HT7 receptor expressed in CHO cell membranes after 120 mins by TopCount scintillation counting metho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464866(CHEMBL4278933)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]LSD from recombinant human 5-HT7 receptor expressed in CHO cell membranes after 120 mins by TopCount scintillation counting metho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464864(CHEMBL4286174)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]LSD from recombinant human 5-HT7 receptor expressed in CHO cell membranes after 120 mins by TopCount scintillation counting metho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50452372(CHEMBL4204665)copy SMILEScopy InChI
Affinity DataKi:  1.5nMAssay Description:Binding affinity to 5-HT1A receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464859(CHEMBL4289361)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Binding affinity to 5-HT1A receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464858(CHEMBL4294077)copy SMILEScopy InChI
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]LSD from recombinant human 5-HT7 receptor expressed in CHO cell membranes after 120 mins by TopCount scintillation counting metho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464856(CHEMBL4288120)copy SMILEScopy InChI
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]LSD from recombinant human 5-HT7 receptor expressed in CHO cell membranes after 120 mins by TopCount scintillation counting metho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464867(CHEMBL4289783)copy SMILEScopy InChI
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]LSD from recombinant human 5-HT7 receptor expressed in CHO cell membranes after 120 mins by TopCount scintillation counting metho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464863(CHEMBL4285796)copy SMILEScopy InChI
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HEK293 cell membranes after 60 mins by TopCount scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464866(CHEMBL4278933)copy SMILEScopy InChI
Affinity DataKi:  8.10nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HEK293 cell membranes after 60 mins by TopCount scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50400902(1-(2-(2,4-dimethylphenylsulfanyl)phenyl)piperazine...)copy SMILEScopy InChI
Affinity DataKi:  9.5nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HEK293 cell membranes after 60 mins by TopCount scintillation count...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464865(CHEMBL4289605)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement of [3H]LSD from recombinant human 5-HT7 receptor expressed in CHO cell membranes after 120 mins by TopCount scintillation counting metho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464864(CHEMBL4286174)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HEK293 cell membranes after 60 mins by TopCount scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464856(CHEMBL4288120)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HEK293 cell membranes after 60 mins by TopCount scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464857(CHEMBL4277476)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HEK293 cell membranes after 60 mins by TopCount scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464858(CHEMBL4294077)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HEK293 cell membranes after 60 mins by TopCount scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464859(CHEMBL4289361)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Inhibition of serotonin reuptake in SERT (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50400902(1-(2-(2,4-dimethylphenylsulfanyl)phenyl)piperazine...)copy SMILEScopy InChI
Affinity DataKi:  26nMAssay Description:Displacement of [3H]LSD from recombinant human 5-HT7 receptor expressed in CHO cell membranes after 120 mins by TopCount scintillation counting metho...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50150105(CHEMBL124069 | [2-(6-Fluoro-chroman-8-yloxy)-ethyl...)copy SMILEScopy InChI
Affinity DataKi:  27nMAssay Description:Binding affinity to 5-HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464867(CHEMBL4289783)copy SMILEScopy InChI
Affinity DataKi:  28nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HEK293 cell membranes after 60 mins by TopCount scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464867(CHEMBL4289783)copy SMILEScopy InChI
Affinity DataKi:  28nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor (unknown origin) in cerebral cortex membranes after 60 mins by TopCount scintillation counting ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464865(CHEMBL4289605)copy SMILEScopy InChI
Affinity DataKi:  62nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in HEK293 cell membranes after 60 mins by TopCount scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50452372(CHEMBL4204665)copy SMILEScopy InChI
Affinity DataKi:  195nMAssay Description:Inhibition of serotonin reuptake in SERT (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50400902(1-(2-(2,4-dimethylphenylsulfanyl)phenyl)piperazine...)copy SMILEScopy InChI
Affinity DataIC50: 2.90nMAssay Description:Inhibition of [3H]serotonin reuptake in rat brain synaptosomes SERT after 15 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464864(CHEMBL4286174)copy SMILEScopy InChI
Affinity DataIC50: 7.60nMAssay Description:Inhibition of [3H]serotonin reuptake in rat brain synaptosomes SERT after 15 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464856(CHEMBL4288120)copy SMILEScopy InChI
Affinity DataIC50: 9.40nMAssay Description:Inhibition of [3H]serotonin reuptake in rat brain synaptosomes SERT after 15 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464857(CHEMBL4277476)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of [3H]serotonin reuptake in rat brain synaptosomes SERT after 15 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464867(CHEMBL4289783)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of [3H]serotonin reuptake in rat brain synaptosomes SERT after 15 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464865(CHEMBL4289605)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of [3H]serotonin reuptake in rat brain synaptosomes SERT after 15 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464866(CHEMBL4278933)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Inhibition of [3H]serotonin reuptake in rat brain synaptosomes SERT after 15 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464858(CHEMBL4294077)copy SMILEScopy InChI
Affinity DataIC50: 96nMAssay Description:Inhibition of [3H]serotonin reuptake in rat brain synaptosomes SERT after 15 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464861(CHEMBL4291322)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of [3H]serotonin reuptake in rat brain synaptosomes SERT after 15 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464870(CHEMBL4279099)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of [3H]serotonin reuptake in rat brain synaptosomes SERT after 15 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464863(CHEMBL4285796)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibition of [3H]serotonin reuptake in rat brain synaptosomes SERT after 15 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464868(CHEMBL4277854)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of [3H]serotonin reuptake in rat brain synaptosomes SERT after 15 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464855(CHEMBL4283479)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Inhibition of [3H]serotonin reuptake in rat brain synaptosomes SERT after 15 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464871(CHEMBL4279592)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Inhibition of [3H]serotonin reuptake in rat brain synaptosomes SERT after 15 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464862(CHEMBL4288753)copy SMILEScopy InChI
Affinity DataIC50: 590nMAssay Description:Inhibition of [3H]serotonin reuptake in rat brain synaptosomes SERT after 15 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464869(CHEMBL4278094)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of [3H]serotonin reuptake in rat brain synaptosomes SERT after 15 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464860(CHEMBL4294729)copy SMILEScopy InChI
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of [3H]serotonin reuptake in rat brain synaptosomes SERT after 15 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Shanghai Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50464867(CHEMBL4289783)copy SMILEScopy InChI
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of human ERG expressed in CHO-K1 cells assessed as reduction in tail current amplitude at -80 mV holding potential after 2 mins by path cl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5WP7PubMed