Compile Data Set for Download or QSAR
Found 20 Enz. Inhib. hit(s) with all data for entry = 50003102
TargetAurora kinase A(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467014(CHEMBL4279747)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using TAMRA-PKAtide as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetAurora kinase A(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467013(CHEMBL4290876)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using TAMRA-PKAtide as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetAurora kinase B(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467019(CHEMBL4277642)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant Aurora B (unknown origin) using TAMRA-PKAtide as substrate after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetAurora kinase B(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467014(CHEMBL4279747)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant Aurora B (unknown origin) using TAMRA-PKAtide as substrate after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetAurora kinase A(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467019(CHEMBL4277642)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using TAMRA-PKAtide as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetAurora kinase B(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467013(CHEMBL4290876)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of recombinant Aurora B (unknown origin) using TAMRA-PKAtide as substrate after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetAurora kinase A(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467017(CHEMBL4284087)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using TAMRA-PKAtide as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetAurora kinase B(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467020(CHEMBL4288081)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant Aurora B (unknown origin) using TAMRA-PKAtide as substrate after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetAurora kinase A(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467020(CHEMBL4288081)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using TAMRA-PKAtide as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetAurora kinase B(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467015(CHEMBL4289877)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Inhibition of recombinant Aurora B (unknown origin) using TAMRA-PKAtide as substrate after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetAurora kinase A(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467015(CHEMBL4289877)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using TAMRA-PKAtide as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetAurora kinase B(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467017(CHEMBL4284087)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Inhibition of recombinant Aurora B (unknown origin) using TAMRA-PKAtide as substrate after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetAurora kinase B(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Inhibition of recombinant Aurora B (unknown origin) using TAMRA-PKAtide as substrate after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetAurora kinase B(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467012(CHEMBL4286456)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of recombinant Aurora B (unknown origin) using TAMRA-PKAtide as substrate after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetAurora kinase B(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467016(CHEMBL4284263)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of recombinant Aurora B (unknown origin) using TAMRA-PKAtide as substrate after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetAurora kinase A(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467016(CHEMBL4284263)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using TAMRA-PKAtide as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetAurora kinase A(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467012(CHEMBL4286456)copy SMILEScopy InChI
Affinity DataIC50: 95nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using TAMRA-PKAtide as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetAurora kinase A(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)copy SMILEScopy InChI
Affinity DataIC50: 127nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using TAMRA-PKAtide as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetAurora kinase B(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467018(CHEMBL4292830)copy SMILEScopy InChI
Affinity DataIC50: 417nMAssay Description:Inhibition of recombinant Aurora B (unknown origin) using TAMRA-PKAtide as substrate after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed
TargetAurora kinase A(Homo sapiens (Human))
MTA-SE Pathobiochemistry Research Group

Curated by ChEMBL
LigandPNGBDBM50467018(CHEMBL4292830)copy SMILEScopy InChI
Affinity DataIC50: 827nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) using TAMRA-PKAtide as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44SZXPubMed