Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with all data for entry = 50003228
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Daegu-Gyeongbuk Medical Innovation Foundation (DGMIF)

Curated by ChEMBL
LigandPNGBDBM25117(AG-013736 | AXITINIB | N-methyl-2-({3-[(E)-2-(pyri...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Inhibition of VEGFR3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8WZZPubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Daegu-Gyeongbuk Medical Innovation Foundation (DGMIF)

Curated by ChEMBL
LigandPNGBDBM25117(AG-013736 | AXITINIB | N-methyl-2-({3-[(E)-2-(pyri...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8WZZPubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Daegu-Gyeongbuk Medical Innovation Foundation (DGMIF)

Curated by ChEMBL
LigandPNGBDBM25117(AG-013736 | AXITINIB | N-methyl-2-({3-[(E)-2-(pyri...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Inhibition of VEGFR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8WZZPubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Daegu-Gyeongbuk Medical Innovation Foundation (DGMIF)

Curated by ChEMBL
LigandPNGBDBM26474(5-({4-[(2,3-dimethyl-2H-indazol-6-yl)(methyl)amino...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of GST-tagged human VEGFR2 C-terminal domain using (biotin-aminohexyl-EEEEYFELVAKKKK-NH2 substrate incubated for 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8WZZPubMedDrugBank