Compile Data Set for Download or QSAR
Found 103 Enz. Inhib. hit(s) with all data for entry = 50003254
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468579(CHEMBL4287262)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468579(CHEMBL4287262)copy SMILEScopy InChI
Affinity DataIC50: 186nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50452662(CHEMBL4208737)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50452662(CHEMBL4208737)copy SMILEScopy InChI
Affinity DataIC50: 234nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM199181(4-[(4-Carbamoylcyclohexyl)oxy]cyclohexane-1-carbox...)copy SMILEScopy InChI
Affinity DataIC50: 330nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM199181(4-[(4-Carbamoylcyclohexyl)oxy]cyclohexane-1-carbox...)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) R931A mutant expressed in Escherichia coli Rosetta2 (DE3) Rosetta2 (DE3) usin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468581(CHEMBL4287655)copy SMILEScopy InChI
Affinity DataIC50: 710nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468581(CHEMBL4287655)copy SMILEScopy InChI
Affinity DataIC50: 710nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468593(CHEMBL4277717)copy SMILEScopy InChI
Affinity DataIC50: 720nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468593(CHEMBL4277717)copy SMILEScopy InChI
Affinity DataIC50: 724nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468581(CHEMBL4287655)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of ARTD10 (unknown origin)-induced cell death expressed in human HeLa cells after 10 days by methylene blue staining based colony formatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468583(CHEMBL4277025)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468583(CHEMBL4277025)copy SMILEScopy InChI
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468578(CHEMBL4285656)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468592(CHEMBL4283907)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468592(CHEMBL4283907)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468578(CHEMBL4285656)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468594(CHEMBL3278113)copy SMILEScopy InChI
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468585(CHEMBL4278641)copy SMILEScopy InChI
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468585(CHEMBL4278641)copy SMILEScopy InChI
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM199181(4-[(4-Carbamoylcyclohexyl)oxy]cyclohexane-1-carbox...)copy SMILEScopy InChI
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of ARTD10 (unknown origin)-induced cell death expressed in human HeLa cells after 10 days by methylene blue staining based colony formatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468580(CHEMBL4294485)copy SMILEScopy InChI
Affinity DataIC50: 1.38E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468587(CHEMBL4289980)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468594(CHEMBL3278113)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468580(CHEMBL4294485)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468587(CHEMBL4289980)copy SMILEScopy InChI
Affinity DataIC50: 1.45E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468586(CHEMBL4277166)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468586(CHEMBL4277166)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468582(CHEMBL4279332)copy SMILEScopy InChI
Affinity DataIC50: 1.74E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468582(CHEMBL4279332)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468595(CHEMBL4293979)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468595(CHEMBL4293979)copy SMILEScopy InChI
Affinity DataIC50: 1.95E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468589(CHEMBL4293554)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468589(CHEMBL4293554)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50452662(CHEMBL4208737)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of ARTD10 (unknown origin)-induced cell death expressed in human HeLa cells after 10 days by methylene blue staining based colony formatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468597(CHEMBL4293771)copy SMILEScopy InChI
Affinity DataIC50: 2.19E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468597(CHEMBL4293771)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468579(CHEMBL4287262)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of N-terminal His-tagged human ARTD7 (482 to 678 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 3 h...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50340090(4-methoxybenzamide | CHEMBL449635)copy SMILEScopy InChI
Affinity DataIC50: 2.75E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50340090(4-methoxybenzamide | CHEMBL449635)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50452662(CHEMBL4208737)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of N-terminal His-tagged human ARTD7 (482 to 678 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 3 h...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50452670(CHEMBL4203858)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50452670(CHEMBL4203858)copy SMILEScopy InChI
Affinity DataIC50: 3.31E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468588(CHEMBL4294759)copy SMILEScopy InChI
Affinity DataIC50: 3.39E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468588(CHEMBL4294759)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468591(CHEMBL4286555)copy SMILEScopy InChI
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468591(CHEMBL4286555)copy SMILEScopy InChI
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP16(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM199181(4-[(4-Carbamoylcyclohexyl)oxy]cyclohexane-1-carbox...)copy SMILEScopy InChI
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of N-terminal His-tagged human ARTD15 (1 to 280 residues) expressed in Escherichia coli Rosetta2 (DE3) after 24 hrs in presence of NAD+More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468596(CHEMBL4282106)copy SMILEScopy InChI
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))
University of Oulu

Curated by ChEMBL
LigandPNGBDBM50468596(CHEMBL4282106)copy SMILEScopy InChI
Affinity DataIC50: 4.57E+3nMAssay Description:Inhibition of C-terminal His-tagged human ARTD10 (809 to 1017 residues) expressed in Escherichia coli Rosetta2 (DE3) using SRPK2 as substrate after 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
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