Compile Data Set for Download or QSAR
Found 155 Enz. Inhib. hit(s) with all data for entry = 50003313
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469353(CHEMBL4283353)copy SMILEScopy InChI
Affinity DataKi:  0.430nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469353(CHEMBL4283353)copy SMILEScopy InChI
Affinity DataKi:  3.90nMAssay Description:Inhibition of TYRO3 (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469353(CHEMBL4283353)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Inhibition of FLT3 (unknown origin) using 5'-FAM-KKKKEEIYFFF-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469353(CHEMBL4283353)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Inhibition of AXL (unknown origin) using 5'-FAM-KKKKEEIYFFF-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50055496(CHEMBL3326006)copy SMILEScopy InChI
Affinity DataIC50: 0.350nMAssay Description:Inhibition of N-terminal GST-tagged human FLT3 cytoplasmic domain (564 to 993 end residues) expressed in baculovirus expression system using fluorece...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50055496(CHEMBL3326006)copy SMILEScopy InChI
Affinity DataIC50: 0.460nMAssay Description:Inhibition of N-terminal GST-tagged human MERTK cytoplasmic domain (528 to 999 end residues) expressed in baculovirus expression system using fluorec...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469353(CHEMBL4283353)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibition of N-terminal GST-tagged human MERTK cytoplasmic domain (528 to 999 end residues) expressed in baculovirus expression system using fluorec...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469376(CHEMBL4284541)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of FLT3 (unknown origin) using 5'-FAM-KKKKEEIYFFF-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469360(CHEMBL4289301)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469376(CHEMBL4284541)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469375(CHEMBL4283152)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of FLT3 (unknown origin) using 5'-FAM-KKKKEEIYFFF-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50055496(CHEMBL3326006)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of N-terminal GST-tagged human AXL cytoplasmic domain (464 to 885 end residues) expressed in baculovirus expression system using fluorecen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50055496(CHEMBL3326006)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of N-terminal GST-tagged human TRKA cytoplasmic domain (436 to 790 end residues) expressed in baculovirus expression system using fluorece...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469354(CHEMBL4286701)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469362(CHEMBL4293116)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469353(CHEMBL4283353)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469358(CHEMBL4277564)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469353(CHEMBL4283353)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of N-terminal GST-tagged human FLT3 cytoplasmic domain (564 to 993 end residues) expressed in baculovirus expression system using fluorece...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469372(CHEMBL4280761)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469349(CHEMBL4281432)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469353(CHEMBL4283353)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Inhibition of N-terminal GST-tagged human TYRO3 cytoplasmic domain (453 to 890 end residues) expressed in baculovirus expression system using fluorec...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469370(CHEMBL4291202)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469364(CHEMBL4291006)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:Inhibition of FLT3 (unknown origin) using 5'-FAM-KKKKEEIYFFF-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469354(CHEMBL4286701)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:Inhibition of TYRO3 (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469366(CHEMBL4282624)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469375(CHEMBL4283152)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469368(CHEMBL4284392)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469371(CHEMBL4288009)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469353(CHEMBL4283353)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Inhibition of N-terminal GST-tagged human TRKA cytoplasmic domain (436 to 790 end residues) expressed in baculovirus expression system using fluorece...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469367(CHEMBL4294601)copy SMILEScopy InChI
Affinity DataIC50: 4.10nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469372(CHEMBL4280761)copy SMILEScopy InChI
Affinity DataIC50: 4.30nMAssay Description:Inhibition of TYRO3 (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469357(CHEMBL4287582)copy SMILEScopy InChI
Affinity DataIC50: 4.30nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM308455(US9649309, Compound UNC2541A)copy SMILEScopy InChI
Affinity DataIC50: 4.40nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469358(CHEMBL4277564)copy SMILEScopy InChI
Affinity DataIC50: 4.40nMAssay Description:Inhibition of TYRO3 (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetNT-3 growth factor receptor(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50055496(CHEMBL3326006)copy SMILEScopy InChI
Affinity DataIC50: 4.40nMAssay Description:Inhibition of N-terminal GST-tagged human TRKC cytoplasmic domain (456 to 825 end residues) expressed in baculovirus expression system using fluorece...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469369(CHEMBL4295042)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469359(CHEMBL4288213)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469350(CHEMBL4284846)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469364(CHEMBL4291006)copy SMILEScopy InChI
Affinity DataIC50: 5.20nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469347(CHEMBL4287078)copy SMILEScopy InChI
Affinity DataIC50: 5.20nMAssay Description:Inhibition of MERTK (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetSerine/threonine-protein kinase SIK2(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50055496(CHEMBL3326006)copy SMILEScopy InChI
Affinity DataIC50: 5.80nMAssay Description:Inhibition of N-terminal GST-tagged full length human QIK (1 to 926 end residues) expressed in baculovirus expression system using fluorecence-labele...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50055496(CHEMBL3326006)copy SMILEScopy InChI
Affinity DataIC50: 5.80nMAssay Description:Inhibition of N-terminal GST-tagged human TYRO3 cytoplasmic domain (453 to 890 end residues) expressed in baculovirus expression system using fluorec...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetSTE20-like serine/threonine-protein kinase(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50055496(CHEMBL3326006)copy SMILEScopy InChI
Affinity DataIC50: 6.10nMAssay Description:Inhibition of N-terminal GST-tagged full length human SLK (1 to 1152 end residues) expressed in baculovirus expression system using fluorecence-label...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469377(CHEMBL4279154)copy SMILEScopy InChI
Affinity DataIC50: 6.70nMAssay Description:Inhibition of TYRO3 (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469366(CHEMBL4282624)copy SMILEScopy InChI
Affinity DataIC50: 6.70nMAssay Description:Inhibition of TYRO3 (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469371(CHEMBL4288009)copy SMILEScopy InChI
Affinity DataIC50: 6.90nMAssay Description:Inhibition of TYRO3 (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50055496(CHEMBL3326006)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of N-terminal GST-tagged full length human NuaK1 (1 to 661 end residues) expressed in baculovirus expression system using fluorecence-labe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50055496(CHEMBL3326006)copy SMILEScopy InChI
Affinity DataIC50: 8.20nMAssay Description:Inhibition of N-terminal GST-tagged human KIT cytoplasmic domain (544 to 976 end residues) expressed in baculovirus expression system using fluorecen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetNT-3 growth factor receptor(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469353(CHEMBL4283353)copy SMILEScopy InChI
Affinity DataIC50: 8.40nMAssay Description:Inhibition of N-terminal GST-tagged human TRKC cytoplasmic domain (456 to 825 end residues) expressed in baculovirus expression system using fluorece...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
UNC Eshelman School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50469360(CHEMBL4289301)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of TYRO3 (unknown origin) using 5'-FAM-EFPIYDFLPAKKK-CONH2 as substrate after 180 mins by MCE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K076ZKPubMed
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