Compile Data Set for Download or QSAR
Found 38 Enz. Inhib. hit(s) with all data for entry = 50003450
TargetGastrin/cholecystokinin type B receptor(MOUSE)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471066(CHEMBL415936)copy SMILEScopy InChI
Affinity DataKi:  0.741nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50213845(CHEMBL14557)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471075(CHEMBL299540)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471067(CHEMBL298521)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471065(CHEMBL296167)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471076(CHEMBL299387)copy SMILEScopy InChI
Affinity DataKi:  3.90nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471072(CHEMBL53237)copy SMILEScopy InChI
Affinity DataKi:  4.10nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471068(CHEMBL298551)copy SMILEScopy InChI
Affinity DataKi:  4.5nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50421390(CHEMBL24313)copy SMILEScopy InChI
Affinity DataKi:  5.20nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471071(CHEMBL297480)copy SMILEScopy InChI
Affinity DataKi:  5.40nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471073(CHEMBL301777)copy SMILEScopy InChI
Affinity DataKi:  7.60nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471064(CHEMBL301810)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471077(CHEMBL280248)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471070(CHEMBL298861)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471062(CHEMBL300456)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471069(CHEMBL53129)copy SMILEScopy InChI
Affinity DataKi:  339nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471063(CHEMBL301095)copy SMILEScopy InChI
Affinity DataKi:  537nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471064(CHEMBL301810)copy SMILEScopy InChI
Affinity DataKi:  851nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471074(CHEMBL301740)copy SMILEScopy InChI
Affinity DataKi:  891nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471072(CHEMBL53237)copy SMILEScopy InChI
Affinity DataKi:  891nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471076(CHEMBL299387)copy SMILEScopy InChI
Affinity DataKi:  912nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471075(CHEMBL299540)copy SMILEScopy InChI
Affinity DataKi:  1.29E+3nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50421390(CHEMBL24313)copy SMILEScopy InChI
Affinity DataKi:  1.48E+3nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471065(CHEMBL296167)copy SMILEScopy InChI
Affinity DataKi:  2.09E+3nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471067(CHEMBL298521)copy SMILEScopy InChI
Affinity DataKi:  2.24E+3nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471068(CHEMBL298551)copy SMILEScopy InChI
Affinity DataKi:  2.57E+3nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471062(CHEMBL300456)copy SMILEScopy InChI
Affinity DataKi:  2.82E+3nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471078(CHEMBL52740)copy SMILEScopy InChI
Affinity DataKi:  2.88E+3nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471070(CHEMBL298861)copy SMILEScopy InChI
Affinity DataKi:  3.16E+3nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471066(CHEMBL415936)copy SMILEScopy InChI
Affinity DataKi:  3.31E+3nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471077(CHEMBL280248)copy SMILEScopy InChI
Affinity DataKi:  3.39E+3nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471069(CHEMBL53129)copy SMILEScopy InChI
Affinity DataKi:  3.55E+3nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50213845(CHEMBL14557)copy SMILEScopy InChI
Affinity DataKi:  3.63E+3nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471071(CHEMBL297480)copy SMILEScopy InChI
Affinity DataKi:  3.80E+3nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471073(CHEMBL301777)copy SMILEScopy InChI
Affinity DataKi:  7.41E+3nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471074(CHEMBL301740)copy SMILEScopy InChI
Affinity DataKi:  8.13E+3nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471063(CHEMBL301095)copy SMILEScopy InChI
Affinity DataKi:  8.32E+3nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471078(CHEMBL52740)copy SMILEScopy InChI
Affinity DataKi:  1.17E+4nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FR6PubMed