TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University of California - Irvine
Curated by ChEMBL
University of California - Irvine
Curated by ChEMBL
Affinity DataKi: 0.0600nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat brain homogenate by scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University of California - Irvine
Curated by ChEMBL
University of California - Irvine
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in Sprague-Dawley rat brain homogenate after 75 mins by scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University of California - Irvine
Curated by ChEMBL
University of California - Irvine
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain homogenateMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University of California - Irvine
Curated by ChEMBL
University of California - Irvine
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat brain homogenate by scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
University of California - Irvine
Curated by ChEMBL
University of California - Irvine
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in Sprague-Dawley rat brain homogenate after 75 mins by scintillation countingMore data for this Ligand-Target Pair