TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of HIV1 capsid protein binding to fluorescein labeled 3-(5-(3-ethyl-5-(5-methylfuran-2-yl)-1H-pyrazol-1-yl)-1-((6-oxo-1,6-dihydropyridin-3...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of HIV1 capsid protein assembly using 5'-fluorescein-labeled (TG)25 oligonucleotide after 2 hrs by fluorometry-based capsid disassembly as...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of HIV1 capsid protein binding to fluorescein labeled 3-(5-(3-ethyl-5-(5-methylfuran-2-yl)-1H-pyrazol-1-yl)-1-((6-oxo-1,6-dihydropyridin-3...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Inhibition of HIV1 capsid protein assembly using 5'-fluorescein-labeled (TG)25 oligonucleotide after 2 hrs by fluorometry-based capsid disassembly as...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of HIV1 capsid protein assembly using 5'-fluorescein-labeled (TG)25 oligonucleotide after 2 hrs by fluorometry-based capsid disassembly as...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibition of HIV1 capsid protein assembly using 5'-fluorescein-labeled (TG)25 oligonucleotide after 2 hrs by fluorometry-based capsid disassembly as...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of HIV1 capsid protein binding to fluorescein labeled 3-(5-(3-ethyl-5-(5-methylfuran-2-yl)-1H-pyrazol-1-yl)-1-((6-oxo-1,6-dihydropyridin-3...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 61nMAssay Description:Inhibition of HIV1 capsid protein binding to fluorescein labeled 3-(5-(3-ethyl-5-(5-methylfuran-2-yl)-1H-pyrazol-1-yl)-1-((6-oxo-1,6-dihydropyridin-3...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Inhibition of HIV1 capsid protein binding to fluorescein labeled 3-(5-(3-ethyl-5-(5-methylfuran-2-yl)-1H-pyrazol-1-yl)-1-((6-oxo-1,6-dihydropyridin-3...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 88nMAssay Description:Inhibition of HIV1 capsid protein assembly using 5'-fluorescein-labeled (TG)25 oligonucleotide after 2 hrs by fluorometry-based capsid disassembly as...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of HIV1 capsid protein assembly using 5'-fluorescein-labeled (TG)25 oligonucleotide after 2 hrs by fluorometry-based capsid disassembly as...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of HIV1 capsid protein assembly using 5'-fluorescein-labeled (TG)25 oligonucleotide after 2 hrs by fluorometry-based capsid disassembly as...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of HIV1 capsid protein assembly using 5'-fluorescein-labeled (TG)25 oligonucleotide after 2 hrs by fluorometry-based capsid disassembly as...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of HIV1 capsid protein assembly using 5'-fluorescein-labeled (TG)25 oligonucleotide after 2 hrs by fluorometry-based capsid disassembly as...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Inhibition of HIV1 capsid protein assembly using 5'-fluorescein-labeled (TG)25 oligonucleotide after 2 hrs by fluorometry-based capsid disassembly as...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 550nMAssay Description:Inhibition of HIV1 capsid protein binding to fluorescein labeled 3-(5-(3-ethyl-5-(5-methylfuran-2-yl)-1H-pyrazol-1-yl)-1-((6-oxo-1,6-dihydropyridin-3...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 650nMAssay Description:Inhibition of HIV1 capsid protein binding to fluorescein labeled 3-(5-(3-ethyl-5-(5-methylfuran-2-yl)-1H-pyrazol-1-yl)-1-((6-oxo-1,6-dihydropyridin-3...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 690nMAssay Description:Inhibition of HIV1 capsid protein binding to fluorescein labeled 3-(5-(3-ethyl-5-(5-methylfuran-2-yl)-1H-pyrazol-1-yl)-1-((6-oxo-1,6-dihydropyridin-3...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 790nMAssay Description:Inhibition of HIV1 capsid protein assembly using 5'-fluorescein-labeled (TG)25 oligonucleotide after 2 hrs by fluorometry-based capsid disassembly as...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 830nMAssay Description:Inhibition of HIV1 capsid protein assembly using 5'-fluorescein-labeled (TG)25 oligonucleotide after 2 hrs by fluorometry-based capsid disassembly as...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HIV1 capsid protein assembly using 5'-fluorescein-labeled (TG)25 oligonucleotide after 2 hrs by fluorometry-based capsid disassembly as...More data for this Ligand-Target Pair
TargetStructural capsid protein(Human immunodeficiency virus 1)
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Boehringer Ingelheim (Canada) Ltd
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of HIV1 capsid protein assembly using 5'-fluorescein-labeled (TG)25 oligonucleotide after 2 hrs by fluorometry-based capsid disassembly as...More data for this Ligand-Target Pair
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