Compile Data Set for Download or QSAR
Found 43 Enz. Inhib. hit(s) with all data for entry = 50005919
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495426(CHEMBL3108801)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Displacement of H4Ac4 peptide from BRD4 bromodomain-1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495431(CHEMBL3108800)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Displacement of H4Ac4 peptide from CECR2 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetCREB-binding protein(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495426(CHEMBL3108801)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Displacement of H3K56(Ac) peptide from CREBBP bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495426(CHEMBL3108801)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Displacement of H2K9(Ac)K13(Ac)K15(Ac) peptide from BRD9 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495431(CHEMBL3108800)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Displacement of H4Ac4 peptide from BRD4 bromodomain-1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495429(CHEMBL3108781)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Displacement of H4Ac4 peptide from CECR2 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495431(CHEMBL3108800)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Displacement of H2K9(Ac)K13(Ac)K15(Ac) peptide from BRD9 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495428(CHEMBL3110357)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Displacement of H4Ac4 peptide from CECR2 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495428(CHEMBL3110357)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Displacement of H2K9(Ac)K13(Ac)K15(Ac) peptide from BRD9 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetCREB-binding protein(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495431(CHEMBL3108800)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Displacement of H3K56(Ac) peptide from CREBBP bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495425(CHEMBL3110353)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Displacement of H2K9(Ac)K13(Ac)K15(Ac) peptide from BRD9 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetCREB-binding protein(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495430(CHEMBL3108803)copy SMILEScopy InChI
Affinity DataIC50: 631nMAssay Description:Displacement of H3K56(Ac) peptide from CREBBP bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetCREB-binding protein(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495425(CHEMBL3110353)copy SMILEScopy InChI
Affinity DataIC50: 794nMAssay Description:Displacement of H3K56(Ac) peptide from CREBBP bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495430(CHEMBL3108803)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of H4Ac4 peptide from BRD4 bromodomain-1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495430(CHEMBL3108803)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of H2K9(Ac)K13(Ac)K15(Ac) peptide from BRD9 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495425(CHEMBL3110353)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of H4Ac4 peptide from CECR2 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495429(CHEMBL3108781)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+3nMAssay Description:Displacement of H4Ac4 peptide from BRD4 bromodomain-1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetCREB-binding protein(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495429(CHEMBL3108781)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+3nMAssay Description:Displacement of H3K56(Ac) peptide from CREBBP bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495427(CHEMBL1513201)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+3nMAssay Description:Displacement of H2K9(Ac)K13(Ac)K15(Ac) peptide from BRD9 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495429(CHEMBL3108781)copy SMILEScopy InChI
Affinity DataIC50: 1.59E+3nMAssay Description:Displacement of H2K9(Ac)K13(Ac)K15(Ac) peptide from BRD9 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetCREB-binding protein(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495427(CHEMBL1513201)copy SMILEScopy InChI
Affinity DataIC50: 1.59E+3nMAssay Description:Displacement of H3K56(Ac) peptide from CREBBP bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495427(CHEMBL1513201)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Displacement of H4Ac4 peptide from BRD4 bromodomain-1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495427(CHEMBL1513201)copy SMILEScopy InChI
Affinity DataIC50: 3.16E+3nMAssay Description:Displacement of H4Ac4 peptide from CECR2 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495425(CHEMBL3110353)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+3nMAssay Description:Displacement of H4Ac4 peptide from BRD4 bromodomain-1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495432(CHEMBL3108806)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+3nMAssay Description:Displacement of H4Ac4 peptide from CECR2 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495428(CHEMBL3110357)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+3nMAssay Description:Displacement of H4Ac4 peptide from BRD4 bromodomain-1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetCREB-binding protein(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495432(CHEMBL3108806)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+3nMAssay Description:Displacement of H3K56(Ac) peptide from CREBBP bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetCREB-binding protein(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495428(CHEMBL3110357)copy SMILEScopy InChI
Affinity DataIC50: 1.58E+4nMAssay Description:Displacement of H3K56(Ac) peptide from CREBBP bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495430(CHEMBL3108803)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Displacement of H4Ac4 peptide from CECR2 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495432(CHEMBL3108806)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Displacement of H4Ac4 peptide from BRD4 bromodomain-1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495426(CHEMBL3108801)copy SMILEScopy InChI
Affinity DataIC50: 2.51E+4nMAssay Description:Displacement of H4Ac4 peptide from CECR2 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495432(CHEMBL3108806)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from TIF1alpha bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495429(CHEMBL3108781)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from BAZ2B bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495432(CHEMBL3108806)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from BAZ2B bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetProtein polybromo-1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495432(CHEMBL3108806)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from PB1-5 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetProtein polybromo-1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495427(CHEMBL1513201)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from PB1-5 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetProtein polybromo-1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495428(CHEMBL3110357)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from PB1-5 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495427(CHEMBL1513201)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from TIF1alpha bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495429(CHEMBL3108781)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from TIF1alpha bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495428(CHEMBL3110357)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from TIF1alpha bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495428(CHEMBL3110357)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from BAZ2B bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetBromodomain adjacent to zinc finger domain protein 2B(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495427(CHEMBL1513201)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from BAZ2B bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed
TargetProtein polybromo-1(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50495429(CHEMBL3108781)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of H3K14(Ac) peptide from PB1-5 bromodomain (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13PDPubMed