TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Inhibition of [3H]-9-cis-RA binding to Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 7.40nMAssay Description:Inhibition of [3H]-9-cis-RA binding to Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2988631PubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2988631PubMedDrugBank
MMDB
PDB
![3D 3D](/images/Docked_3d.png)
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 8.40nMAssay Description:Inhibition of [3H]-9-cis-RA binding to Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2988631PubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2988631PubMedDrugBank
MMDB
PDB
![3D 3D](/images/Docked_3d.png)
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 9.30nMAssay Description:Inhibition of [3H]-9-cis-RA binding to Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 9.30nMAssay Description:Inhibition of [3H]-9-cis-RA binding to Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 10.2nMAssay Description:Inhibition of [3H]-9-cis-RA binding to Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 10.2nMAssay Description:Inhibition of [3H]-9-cis-RA binding to Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Inhibition of [3H]-ATRA binding to Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Inhibition of [3H]-9-cis-RA binding to Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2988631PubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2988631PubMedDrugBank
MMDB
PDB
![3D 3D](/images/Docked_3d.png)
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Inhibition of [3H]-ATRA binding to Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Inhibition of [3H]-ATRA binding to Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of [3H]-ATRA binding to Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Inhibition of [3H]-ATRA binding to Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 64nMAssay Description:Inhibition of [3H]-ATRA binding to Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 64nMAssay Description:Inhibition of [3H]-ATRA binding to Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Inhibition of [3H]-ATRA binding to Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 124nMAssay Description:Inhibition of [3H]-ATRA binding to Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 124nMAssay Description:Inhibition of [3H]-ATRA binding to Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 187nMAssay Description:Inhibition of [3H]-ATRA binding to Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 288nMAssay Description:Inhibition of [3H]-9-cis-RA binding to Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 350nMAssay Description:Inhibition of [3H]-9-cis-RA binding to Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 881nMAssay Description:Inhibition of [3H]-9-cis-RA binding to Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 134nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 105nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 52nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 200nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2988631PubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2988631PubMedDrugBank
MMDB
PDB
![3D 3D](/images/Docked_3d.png)
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 77nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 304nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 316nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2988631PubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2988631PubMedDrugBank
MMDB
PDB
![3D 3D](/images/Docked_3d.png)
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 1.23E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 1.39E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 65nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-beta(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 87nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoid X receptor RXR betaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 16nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 1.08E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoid X receptor RXR alphaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 24nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 563nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 74nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 219nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2988631PubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2988631PubMedDrugBank
MMDB
PDB
![3D 3D](/images/Docked_3d.png)
TargetRetinoic acid receptor beta(Homo sapiens (Human))
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Ligand Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 24nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
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