Found 12 Enz. Inhib. hit(s) with all data for entry = 50007722 TargetSerine protease hepsin(Homo sapiens (Human))
Universidade Federal de Pernambuco
Curated by ChEMBL
Universidade Federal de Pernambuco
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Inhibition of recombinant human hepsin preincubated for 30 mins followed by Boc-QLR-AMC substrate addition by fluorescence assayMore data for this Ligand-Target Pair
TargetSerine protease hepsin(Homo sapiens (Human))
Universidade Federal de Pernambuco
Curated by ChEMBL
Universidade Federal de Pernambuco
Curated by ChEMBL
Affinity DataKi: 0.670nMAssay Description:Inhibition of recombinant human hepsin preincubated for 30 mins followed by Boc-QLR-AMC substrate addition by fluorescence assayMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Universidade Federal de Pernambuco
Curated by ChEMBL
Universidade Federal de Pernambuco
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Inhibition of recombinant human matriptase preincubated for 30 mins followed by Boc-QLR-AMC substrate addition by fluorescence assayMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Universidade Federal de Pernambuco
Curated by ChEMBL
Universidade Federal de Pernambuco
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Inhibition of recombinant human matriptase preincubated for 30 mins followed by Boc-QLR-AMC substrate addition by fluorescence assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor activator(Homo sapiens (Human))
Universidade Federal de Pernambuco
Curated by ChEMBL
Universidade Federal de Pernambuco
Curated by ChEMBL
Affinity DataKi: 3.70nMAssay Description:Inhibition of recombinant HGFA serine protease domain (unknown origin) preincubated for 30 mins followed by Boc-QLR-AMC substrate addition by fluores...More data for this Ligand-Target Pair
TargetHepatocyte growth factor activator(Homo sapiens (Human))
Universidade Federal de Pernambuco
Curated by ChEMBL
Universidade Federal de Pernambuco
Curated by ChEMBL
Affinity DataKi: 7.20nMAssay Description:Inhibition of recombinant HGFA serine protease domain (unknown origin) preincubated for 30 mins followed by Boc-QLR-AMC substrate addition by fluores...More data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Inhibition of recombinant factor 10a (unknown origin) preincubated for 30 mins followed by chromogenic substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 447nMAssay Description:Inhibition of recombinant factor 10a (unknown origin) preincubated for 30 mins followed by chromogenic substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.62E+3nMAssay Description:Inhibition of recombinant thrombin (unknown origin) preincubated for 30 mins followed by chromogenic substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.95E+3nMAssay Description:Inhibition of recombinant thrombin (unknown origin) preincubated for 30 mins followed by chromogenic substrate addition by fluorescence assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Universidade Federal de Pernambuco
Curated by ChEMBL
Universidade Federal de Pernambuco
Curated by ChEMBL
Affinity DataIC50: 73nMAssay Description:Inhibition of HDAC1 (unknown origin) using Ac-peptide as substrate pretreated for 15 mins followed by substrate addition and measured after 60 mins b...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universidade Federal de Pernambuco
Curated by ChEMBL
Universidade Federal de Pernambuco
Curated by ChEMBL
Affinity DataIC50: 97nMAssay Description:Inhibition of SRC (unknown origin) by Z'-LYTE assayMore data for this Ligand-Target Pair
