Compile Data Set for Download or QSAR
Found 12 Enz. Inhib. hit(s) with all data for entry = 50008003
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cullgen Inc.

Curated by ChEMBL
LigandPNGBDBM50514785(CHEMBL4443903)copy SMILEScopy InChI
Affinity DataKd:  2.40nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) by KINOMEscan assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD1511PubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cullgen Inc.

Curated by ChEMBL
LigandPNGBDBM50514786(CHEMBL4541406)copy SMILEScopy InChI
Affinity DataKd:  14nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) V600E mutant by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD1511PubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cullgen Inc.

Curated by ChEMBL
LigandPNGBDBM50514787(CHEMBL4449322)copy SMILEScopy InChI
Affinity DataKd:  7.30nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) V600E mutant by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD1511PubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cullgen Inc.

Curated by ChEMBL
LigandPNGBDBM50514788(CHEMBL4440761)copy SMILEScopy InChI
Affinity DataKd:  2.70nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) V600E mutant by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD1511PubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cullgen Inc.

Curated by ChEMBL
LigandPNGBDBM50457446(CHEMBL4212692)copy SMILEScopy InChI
Affinity DataKd:  0.330nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) V600E mutant by KINOMEscan assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cullgen Inc.

Curated by ChEMBL
LigandPNGBDBM50396483(PLX-4032 | RG 7204 | Ro 5185426 | US10570155, Vemu...)copy SMILEScopy InChI
Affinity DataKd:  58nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) V600E mutant by KINOMEscan assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cullgen Inc.

Curated by ChEMBL
LigandPNGBDBM50514788(CHEMBL4440761)copy SMILEScopy InChI
Affinity DataKd:  2.60nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD1511PubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cullgen Inc.

Curated by ChEMBL
LigandPNGBDBM50457446(CHEMBL4212692)copy SMILEScopy InChI
Affinity DataKd:  0.370nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) by KINOMEscan assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cullgen Inc.

Curated by ChEMBL
LigandPNGBDBM50514786(CHEMBL4541406)copy SMILEScopy InChI
Affinity DataKd:  9.5nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD1511PubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cullgen Inc.

Curated by ChEMBL
LigandPNGBDBM50514785(CHEMBL4443903)copy SMILEScopy InChI
Affinity DataKd:  2nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) V600E mutant by KINOMEscan assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD1511PubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cullgen Inc.

Curated by ChEMBL
LigandPNGBDBM50514787(CHEMBL4449322)copy SMILEScopy InChI
Affinity DataKd:  5.10nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD1511PubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Cullgen Inc.

Curated by ChEMBL
LigandPNGBDBM50396483(PLX-4032 | RG 7204 | Ro 5185426 | US10570155, Vemu...)copy SMILEScopy InChI
Affinity DataKd:  51nMAssay Description:Binding affinity to DNA-tagged BRAF (unknown origin) by KINOMEscan assayMore data for this Ligand-Target Pair