TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by ChEMBL
Bristol-Myers Squibb
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Inhibition of His6 tagged human FKBP12 expressed in Escherichia coli BL21(DE3) cells using succinylALPF-p-nitroanilide as substrate by fluorescence p...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity to mu opioid receptor (unknown origin) expressed in HEK cells at pH 7.4More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Binding affinity to mu opioid receptor (unknown origin) expressed in HEK cells at pH 6.5More data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Binding affinity to delta opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Binding affinity to mu opioid receptor (unknown origin) expressed in HEK cells at pH 5.5More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity to mu opioid receptor (unknown origin) expressed in HEK cells at pH 7.4More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by ChEMBL
Bristol-Myers Squibb
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Inhibition of His6 tagged human FKBP12 expressed in Escherichia coli BL21(DE3) cells using succinylALPF-p-nitroanilide as substrate by fluorescence p...More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Inhibition of human androgen receptorMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Inhibition of human androgen receptorMore data for this Ligand-Target Pair
TargetGenome polyprotein(Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Bristol-Myers Squibb
Curated by ChEMBL
Bristol-Myers Squibb
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of HCV NS3 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Binding affinity to delta opioid receptor (unknown origin)More data for this Ligand-Target Pair
TargetGenome polyprotein(Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Bristol-Myers Squibb
Curated by ChEMBL
Bristol-Myers Squibb
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of HCV NS3 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Binding affinity to delta opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Binding affinity to delta opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 158nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 158nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 251nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 251nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 310nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 398nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 490nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Inhibition of thrombin (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 587nMAssay Description:Binding affinity to delta opioid receptor (unknown origin)More data for this Ligand-Target Pair
TargetGenome polyprotein(Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Bristol-Myers Squibb
Curated by ChEMBL
Bristol-Myers Squibb
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Inhibition of HCV NS3 proteaseMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by ChEMBL
Bristol-Myers Squibb
Curated by ChEMBL
Affinity DataKi: 870nMAssay Description:Inhibition of His6 tagged human FKBP12 expressed in Escherichia coli BL21(DE3) cells using succinylALPF-p-nitroanilide as substrate by fluorescence p...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by ChEMBL
Bristol-Myers Squibb
Curated by ChEMBL
Affinity DataKi: 4.00E+3nMAssay Description:Inhibition of His6 tagged human FKBP12 expressed in Escherichia coli BL21(DE3) cells using succinylALPF-p-nitroanilide as substrate by fluorescence p...More data for this Ligand-Target Pair
Affinity DataKi: 2.40E+4nMAssay Description:Competitive inhibition of trypanosoma cruzi trypanothione reductaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.80E+4nMAssay Description:Inhibition of steroid sulfatase (unknown origin) at pH 8.8More data for this Ligand-Target Pair
Affinity DataKi: 2.80E+4nMAssay Description:Competitive inhibition of trypanosoma cruzi trypanothione reductaseMore data for this Ligand-Target Pair
Affinity DataKi: 5.70E+4nMAssay Description:Inhibition of steroid sulfatase (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 7.30E+4nMAssay Description:Inhibition of steroid sulfatase (unknown origin) at pH 7More data for this Ligand-Target Pair
Affinity DataKi: 8.20E+4nMAssay Description:Inhibition of steroid sulfatase (unknown origin) at pH 7More data for this Ligand-Target Pair
Affinity DataKi: 8.40E+4nMAssay Description:Competitive inhibition of trypanosoma cruzi trypanothione reductaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.47E+5nMAssay Description:Inhibition of steroid sulfatase (unknown origin) at pH 8.8More data for this Ligand-Target Pair
Affinity DataKi: 3.50E+5nMAssay Description:Inhibition of steroid sulfatase (unknown origin) at pH 7More data for this Ligand-Target Pair
Affinity DataKi: 6.00E+5nMAssay Description:Inhibition of steroid sulfatase (unknown origin)More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by ChEMBL
Bristol-Myers Squibb
Curated by ChEMBL
Affinity DataKi: 6.30E+6nMAssay Description:Competitive inhibition of GABA aminotransferase (unknown origin)More data for this Ligand-Target Pair
Target4-aminobutyrate aminotransferase, mitochondrial(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by ChEMBL
Bristol-Myers Squibb
Curated by ChEMBL
Affinity DataKi: 1.10E+7nMAssay Description:Competitive inhibition of GABA aminotransferase (unknown origin)More data for this Ligand-Target Pair
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Bristol-Myers Squibb
Curated by ChEMBL
Bristol-Myers Squibb
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human type 2 5alpha reductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:Inhibition of human 5HT1D expressed in CHO cells by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair