Affinity DataKi: 8.5nMAssay Description:Partial agonist activity at human D1RMore data for this Ligand-Target Pair
Affinity DataKi: 113nMAssay Description:Partial agonist activity at human D1RMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Positive allosteric modulation of human D1R expressed in HEK293 cells assessed as increase in dopamine-induced cAMP accumulation after 60 mins by HTR...More data for this Ligand-Target Pair
Affinity DataEC50: 1.87E+3nMAssay Description:Positive allosteric modulation of D1R (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Affinity DataEC50: 330nMAssay Description:Agonist activity at D2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 56nMAssay Description:Positive allosteric modulation of human D1R expressed in HEK cells assessed as increase in dopamine-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 250nMAssay Description:Positive allosteric modulation of human D1R expressed in HEK cells assessed as increase in dopamine-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 5.80nMAssay Description:Positive allosteric modulation of human D1R expressed in HEK293 cells assessed as increase in dopamine-induced cAMP accumulation after 60 mins by HTR...More data for this Ligand-Target Pair
Affinity DataEC50: 210nMAssay Description:Positive allosteric modulation of human D1R expressed in CHO cells assessed as increase in dopamine-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 460nMAssay Description:Positive allosteric modulation of human D1R expressed in CHO cells assessed as 2-fold increase in dopamine-induced cAMP accumulation preincubated for...More data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Positive allosteric modulation of human D1R expressed in HEK293 cells assessed as increase in dopamine-induced cAMP accumulation after 60 mins by HTR...More data for this Ligand-Target Pair
Affinity DataEC50: 162nMAssay Description:Positive allosteric modulation of rat D1R expressed in HEK293 cells assessed as increase in dopamine-induced cAMP accumulation after 60 mins by HTRF ...More data for this Ligand-Target Pair
Affinity DataEC50: 3.70nMAssay Description:Positive allosteric modulation of human D1R expressed in HEK293 cells assessed as increase in dopamine-induced cAMP accumulation after 60 mins by HTR...More data for this Ligand-Target Pair
Affinity DataEC50: 332nMAssay Description:Positive allosteric modulation of rat D1R expressed in HEK cells assessed as increase in dopamine-induced cAMP accumulation relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Positive allosteric modulation of human D1R expressed in HEK cells assessed as increase in dopamine-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Positive allosteric modulation of human D1R expressed in CHO cells assessed as increase in dopamine-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 165nMAssay Description:Positive allosteric modulation of D1R (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of rat D1R expressed in HEK cells assessed as increase in dopamine-induced cAMP accumulation relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 440nMAssay Description:Positive allosteric modulation of human D1R expressed in CHO cells assessed as 2-fold increase in dopamine-induced cAMP accumulation preincubated for...More data for this Ligand-Target Pair
Affinity DataEC50: 312nMAssay Description:Positive allosteric modulation of mouse D1R expressed in HEK293 cells assessed as increase in dopamine-induced cAMP accumulation after 60 mins by HTR...More data for this Ligand-Target Pair