Compile Data Set for Download or QSAR
Found 16 Enz. Inhib. hit(s) with all data for entry = 50008897
TargetAromatase(Homo sapiens (Human))
University of Coimbra

Curated by ChEMBL
LigandPNGBDBM50135997(CHEMBL3754471)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Competitive irreversible inhibition of human placental microsome aromatase using varying levels of [1beta3H]-androstenedione as substrate measured af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301CWPubMed
TargetAromatase(Homo sapiens (Human))
University of Coimbra

Curated by ChEMBL
LigandPNGBDBM50135997(CHEMBL3754471)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Competitive reversible inhibition of human placental microsome aromatase using varying levels of [1beta3H]-androstenedione as substrate measured afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301CWPubMed
TargetAromatase(Homo sapiens (Human))
University of Coimbra

Curated by ChEMBL
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)copy SMILEScopy InChI
Affinity DataKi:  26nMAssay Description:Competitive inhibition of human placental microsome aromatase using varying levels of [1beta2beta3H]-androstenedione as substrateMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
University of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523404(CHEMBL4575994)copy SMILEScopy InChI
Affinity DataIC50: 55nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301CWPubMed
TargetAromatase(Homo sapiens (Human))
University of Coimbra

Curated by ChEMBL
LigandPNGBDBM50135997(CHEMBL3754471)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301CWPubMed
TargetAromatase(Homo sapiens (Human))
University of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523395(CHEMBL4514728)copy SMILEScopy InChI
Affinity DataIC50: 105nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301CWPubMed
TargetAromatase(Homo sapiens (Human))
University of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523399(CHEMBL4454575)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301CWPubMed
TargetAromatase(Homo sapiens (Human))
University of Coimbra

Curated by ChEMBL
LigandPNGBDBM50135862(CHEMBL3751881)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301CWPubMed
TargetAromatase(Homo sapiens (Human))
University of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523403(CHEMBL4460869)copy SMILEScopy InChI
Affinity DataIC50: 175nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301CWPubMed
TargetAromatase(Homo sapiens (Human))
University of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523400(CHEMBL4520056)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301CWPubMed
TargetAromatase(Homo sapiens (Human))
University of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523396(CHEMBL487113)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301CWPubMed
TargetAromatase(Homo sapiens (Human))
University of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523397(CHEMBL4451962)copy SMILEScopy InChI
Affinity DataIC50: 405nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301CWPubMed
TargetAromatase(Homo sapiens (Human))
University of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523402(CHEMBL4468497)copy SMILEScopy InChI
Affinity DataIC50: 520nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301CWPubMed
TargetAromatase(Homo sapiens (Human))
University of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523398(CHEMBL4564333)copy SMILEScopy InChI
Affinity DataIC50: 560nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301CWPubMed
TargetAromatase(Homo sapiens (Human))
University of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523401(CHEMBL4515880)copy SMILEScopy InChI
Affinity DataIC50: 840nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301CWPubMed
TargetAromatase(Homo sapiens (Human))
University of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523405(CHEMBL4520027)copy SMILEScopy InChI
Affinity DataIC50: 880nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301CWPubMed