Found 6 Enz. Inhib. hit(s) with all data for entry = 50009069 TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
University Health Network
Curated by ChEMBL
University Health Network
Curated by ChEMBL
Affinity DataKd: 2.00E+4nMAssay Description:Inhibition of 8-NBD-cAMP binding to human EPAC1 cAMP binding domain (149 to 318 residues) by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKd: 99nMAssay Description:Displacement of dansylated phenylalanine from human serum albumin by fluorescence assayMore data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
University Health Network
Curated by ChEMBL
University Health Network
Curated by ChEMBL
Affinity DataKd: 7.57E+5nMAssay Description:Binding affinity to human EPAC1 cAMP binding domain (149 to 318 residues) in presence of human serum albumin by [15N-1H]HSQC spectroscopic analysisMore data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
University Health Network
Curated by ChEMBL
University Health Network
Curated by ChEMBL
Affinity DataKd: 1.24E+5nMAssay Description:Binding affinity to human EPAC1 cAMP binding domain (149 to 318 residues) by [15N-1H]HSQC spectroscopic analysisMore data for this Ligand-Target Pair
Affinity DataKd: 230nMAssay Description:Displacement of dansylated arginine from human serum albumin by fluorescence assayMore data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
University Health Network
Curated by ChEMBL
University Health Network
Curated by ChEMBL
Affinity DataKd: 2.00E+4nMAssay Description:Binding affinity to human EPAC1 cAMP binding domain (149 to 318 residues) using aggregate form of compound by [15N-1H]HSQC spectroscopic analysisMore data for this Ligand-Target Pair
