TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 0.130nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of CDK5 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of CDK2/cycE1 (unknown origin) by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 6.40nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of CDK7/CycH/MAT1 (unknown origin) by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of CDK7/CycH/MAT1 (unknown origin) by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of CDK7 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of CDK9 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of CDK7 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q24X5C86PubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q24X5C86PubMedDrugBank
MMDB
PDB
3D Structure (crystal)
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of CDK9 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of CDK7 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of CDK7/CycH/MAT1 (unknown origin) by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of CDK1 (unknown origin) by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 6(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of CDK6 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 97nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of CDK4 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 134nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of CDK5 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 194nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of CDK5 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of CDK2 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair