Compile Data Set for Download or QSAR
Found 56 Enz. Inhib. hit(s) with all data for entry = 50009894
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195608(CPI-455)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of KDM5B (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195608(CPI-455)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of KDM5B (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195608(CPI-455)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195608(CPI-455)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533317(CHEMBL4538785)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533317(CHEMBL4538785)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533308(CHEMBL4444632)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533308(CHEMBL4444632)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5C(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195608(CPI-455)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of KDM5C (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5C(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195608(CPI-455)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of KDM5C (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533309(CHEMBL4464860)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533309(CHEMBL4464860)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195610(KDM inhibitor, 3)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195608(CPI-455)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/20 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195610(KDM inhibitor, 3)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195608(CPI-455)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/20 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM191596(6-isopropyl-5-methyl-7-oxo-4,7-dihydropyrazolo[1,5...)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM191596(6-isopropyl-5-methyl-7-oxo-4,7-dihydropyrazolo[1,5...)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533312(CHEMBL4557175)copy SMILEScopy InChI
Affinity DataIC50: 55nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533312(CHEMBL4557175)copy SMILEScopy InChI
Affinity DataIC50: 55nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195609(CPI-4203)copy SMILEScopy InChI
Affinity DataIC50: 206nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195609(CPI-4203)copy SMILEScopy InChI
Affinity DataIC50: 206nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533315(CHEMBL4520731)copy SMILEScopy InChI
Affinity DataIC50: 214nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533315(CHEMBL4520731)copy SMILEScopy InChI
Affinity DataIC50: 214nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533305(CHEMBL4469878)copy SMILEScopy InChI
Affinity DataIC50: 237nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533305(CHEMBL4469878)copy SMILEScopy InChI
Affinity DataIC50: 237nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50158828(CHEMBL3786528)copy SMILEScopy InChI
Affinity DataIC50: 324nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50158828(CHEMBL3786528)copy SMILEScopy InChI
Affinity DataIC50: 324nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533313(CHEMBL4448240)copy SMILEScopy InChI
Affinity DataIC50: 649nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533313(CHEMBL4448240)copy SMILEScopy InChI
Affinity DataIC50: 649nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533310(CHEMBL4452124)copy SMILEScopy InChI
Affinity DataIC50: 712nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533310(CHEMBL4452124)copy SMILEScopy InChI
Affinity DataIC50: 712nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50158826(CHEMBL3786862)copy SMILEScopy InChI
Affinity DataIC50: 878nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50158826(CHEMBL3786862)copy SMILEScopy InChI
Affinity DataIC50: 878nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533314(CHEMBL4530774)copy SMILEScopy InChI
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533314(CHEMBL4530774)copy SMILEScopy InChI
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195608(CPI-455)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of KDM4C (unknown origin) using ARTKQTAR(KMe3)STGGKAPRKQLA-NovaTagPEG-biotin/2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195608(CPI-455)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of KDM4C (unknown origin) using ARTKQTAR(KMe3)STGGKAPRKQLA-NovaTagPEG-biotin/2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533316(CHEMBL4474445)copy SMILEScopy InChI
Affinity DataIC50: 2.24E+3nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533316(CHEMBL4474445)copy SMILEScopy InChI
Affinity DataIC50: 2.24E+3nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533306(CHEMBL4517696)copy SMILEScopy InChI
Affinity DataIC50: 3.09E+3nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533306(CHEMBL4517696)copy SMILEScopy InChI
Affinity DataIC50: 3.09E+3nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195608(CPI-455)copy SMILEScopy InChI
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of KDM7B (unknown origin) ARTKQTAR(KMe1)STGGKAPRKQLA-NovaTagPEG-biotin/2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195608(CPI-455)copy SMILEScopy InChI
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of KDM7B (unknown origin) ARTKQTAR(KMe1)STGGKAPRKQLA-NovaTagPEG-biotin/2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533307(CHEMBL4460935)copy SMILEScopy InChI
Affinity DataIC50: 8.94E+3nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50533307(CHEMBL4460935)copy SMILEScopy InChI
Affinity DataIC50: 8.94E+3nMAssay Description:Inhibition of KDM5A (unknown origin) using ART(Kme3)QTARKSTGGKAPRKQLA-NovaTagPEG-biotin/1 uM 2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 2B(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195608(CPI-455)copy SMILEScopy InChI
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of KDM2B (unknown origin) using RKSAPATGGV(KMe2)KPHRYRPGTV-NovaTagPEG-biotin/2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 2B(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195608(CPI-455)copy SMILEScopy InChI
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of KDM2B (unknown origin) using RKSAPATGGV(KMe2)KPHRYRPGTV-NovaTagPEG-biotin/2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 3B(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195608(CPI-455)copy SMILEScopy InChI
Affinity DataIC50: 1.53E+4nMAssay Description:Inhibition of KDM3B (unknown origin) using ARTKQTAR(KMe1)STGGKAPRKQLA -NovaTagPEG-biotin/2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
TargetLysine-specific demethylase 3B(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM195608(CPI-455)copy SMILEScopy InChI
Affinity DataIC50: 1.53E+4nMAssay Description:Inhibition of KDM3B (unknown origin) using ARTKQTAR(KMe1)STGGKAPRKQLA -NovaTagPEG-biotin/2-OG as substrate/co-factor by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2MNWPubMed
Displayed 1 to 50 (of 56 total ) | Next | Last >>
Jump to: