Compile Data Set for Download or QSAR
Found 75 Enz. Inhib. hit(s) with all data for entry = 50010508
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50539719(CHEMBL4644434)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50539722(CHEMBL4644572)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50526792(CHEMBL4454044)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50539722(CHEMBL4644572)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in baculovirus infected Sf21 insect cells in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM101536(CHEMBL3128043 | US8530494, 203 | US8530652, 114 | ...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of CDK7/cyclin H/MNAT1 (unknown origin) pre incubated up to 60 mins followed by substrate and ATP additionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50526803(CHEMBL4434871 | US10870651, Compound 101)copy SMILEScopy InChI
Affinity DataIC50: 7.60nMAssay Description:Inhibition of CDK7/cyclin H/MNAT1 (unknown origin) pre incubated up to 60 mins followed by substrate and ATP additionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50526795(CHEMBL4450322)copy SMILEScopy InChI
Affinity DataIC50: 9.70nMAssay Description:Inhibition of CDK7/cyclin H/MNAT1 (unknown origin) pre incubated up to 60 mins followed by substrate and ATP additionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50526794(CHEMBL4303287 | US10787436, Compound I-18)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of CDK7/cyclin H/MNAT1 (unknown origin) pre incubated up to 60 mins followed by substrate and ATP additionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50539720(CHEMBL4648392)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50539718(CHEMBL4643708)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50539709(CHEMBL4649721)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50347389(CHEMBL1801932)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50528814(CHEMBL4436535)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of CDK7/cyclin H/MNAT1 (unknown origin) pre incubated up to 60 mins followed by substrate and ATP additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50539710(CHEMBL4637408)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50539712(CHEMBL4639779)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50526797(Ct-7001 | Ct7001 | ICEC-0942 | ICEC0942 | Samuraci...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50539715(CHEMBL4635439)copy SMILEScopy InChI
Affinity DataIC50: 59nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50539714(CHEMBL4633156)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50539707(CHEMBL4636757)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50528812(CHEMBL4582951)copy SMILEScopy InChI
Affinity DataIC50: 84nMAssay Description:Inhibition of CDK7/cyclin H/MNAT1 (unknown origin) pre incubated up to 60 mins followed by substrate and ATP additionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50526794(CHEMBL4303287 | US10787436, Compound I-18)copy SMILEScopy InChI
Affinity DataIC50: 97nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM7533((2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]am...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin) expressed in baculovirus infected Sf21 insect cells in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50528811(CHEMBL4441405)copy SMILEScopy InChI
Affinity DataIC50: 112nMAssay Description:Inhibition of CDK7/cyclin H/MNAT1 (unknown origin) pre incubated up to 60 mins followed by substrate and ATP additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50526794(CHEMBL4303287 | US10787436, Compound I-18)copy SMILEScopy InChI
Affinity DataIC50: 134nMAssay Description:Inhibition of CDK5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50539721(CHEMBL4635959)copy SMILEScopy InChI
Affinity DataIC50: 148nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50528813(CHEMBL4163879)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 8(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50526794(CHEMBL4303287 | US10787436, Compound I-18)copy SMILEScopy InChI
Affinity DataIC50: 194nMAssay Description:Inhibition of CDK8 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 12(Homo sapiens)
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50528812(CHEMBL4582951)copy SMILEScopy InChI
Affinity DataIC50: 204nMAssay Description:Inhibition of CDK12 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50526794(CHEMBL4303287 | US10787436, Compound I-18)copy SMILEScopy InChI
Affinity DataIC50: 222nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50110178(CHEMBL3603847 | US10787436, Compound I-23)copy SMILEScopy InChI
Affinity DataIC50: 238nMAssay Description:Inhibition of CDK7/cyclin H/MNAT1 (unknown origin) pre incubated up to 60 mins followed by substrate and ATP additionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50539719(CHEMBL4644434)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50526805(CHEMBL4519886)copy SMILEScopy InChI
Affinity DataIC50: 310nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50539713(CHEMBL4646646)copy SMILEScopy InChI
Affinity DataIC50: 320nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM7533((2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]am...)copy SMILEScopy InChI
Affinity DataIC50: 510nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50526797(Ct-7001 | Ct7001 | ICEC-0942 | ICEC0942 | Samuraci...)copy SMILEScopy InChI
Affinity DataIC50: 620nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 13(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50110178(CHEMBL3603847 | US10787436, Compound I-23)copy SMILEScopy InChI
Affinity DataIC50: 628nMAssay Description:Inhibition of CDK13 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50539711(CHEMBL4637421)copy SMILEScopy InChI
Affinity DataIC50: 654nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50526796(CHEMBL4472515)copy SMILEScopy InChI
Affinity DataIC50: 687nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50347389(CHEMBL1801932)copy SMILEScopy InChI
Affinity DataIC50: 880nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 12(Homo sapiens)
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50110178(CHEMBL3603847 | US10787436, Compound I-23)copy SMILEScopy InChI
Affinity DataIC50: 893nMAssay Description:Inhibition of CDK12 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50528812(CHEMBL4582951)copy SMILEScopy InChI
Affinity DataIC50: 914nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50539717(CHEMBL4646538)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50539716(CHEMBL4632793)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50539708(CHEMBL4638833)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50526803(CHEMBL4434871 | US10870651, Compound 101)copy SMILEScopy InChI
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50526797(Ct-7001 | Ct7001 | ICEC-0942 | ICEC0942 | Samuraci...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50526795(CHEMBL4450322)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50526797(Ct-7001 | Ct7001 | ICEC-0942 | ICEC0942 | Samuraci...)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50528812(CHEMBL4582951)copy SMILEScopy InChI
Affinity DataIC50: 2.12E+3nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Lebanese American University

Curated by ChEMBL
LigandPNGBDBM50539721(CHEMBL4635959)copy SMILEScopy InChI
Affinity DataIC50: 2.83E+3nMAssay Description:Inhibition of CDK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C82DT8PubMed
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