Compile Data Set for Download or QSAR
Found 79 Enz. Inhib. hit(s) with all data for entry = 50011073
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50505255(BIIB-074 | BIIB074 | CNV-1014802 | CNV1014802 | GS...)copy SMILEScopy InChI
Affinity DataKi: <1.00E+4nMAssay Description:Inhibition of MAO-A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50505255(BIIB-074 | BIIB074 | CNV-1014802 | CNV1014802 | GS...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of MAO-B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544669(CHEMBL4647249)copy SMILEScopy InChI
Affinity DataIC50: 3.16E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544671(CHEMBL4644347)copy SMILEScopy InChI
Affinity DataIC50: 3.16E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544677(CHEMBL4634692)copy SMILEScopy InChI
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544687(CHEMBL4634823)copy SMILEScopy InChI
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544681(CHEMBL4646446)copy SMILEScopy InChI
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544685(CHEMBL4635537)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544667(CHEMBL4634427)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544666(CHEMBL4644276)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544674(CHEMBL4645734)copy SMILEScopy InChI
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544673(CHEMBL4642930)copy SMILEScopy InChI
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544672(CHEMBL4644773)copy SMILEScopy InChI
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544686(CHEMBL4648552)copy SMILEScopy InChI
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544665(CHEMBL4647983)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544675(CHEMBL4637902)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50505255(BIIB-074 | BIIB074 | CNV-1014802 | CNV1014802 | GS...)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544678(CHEMBL4634636)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544684(CHEMBL4635448)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50505255(BIIB-074 | BIIB074 | CNV-1014802 | CNV1014802 | GS...)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544676(CHEMBL4635121)copy SMILEScopy InChI
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544683(CHEMBL4648908)copy SMILEScopy InChI
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544682(CHEMBL4637843)copy SMILEScopy InChI
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544651(CHEMBL4634172)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544680(CHEMBL4638413)copy SMILEScopy InChI
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544689(CHEMBL4632663)copy SMILEScopy InChI
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544670(CHEMBL4649796)copy SMILEScopy InChI
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetCytochrome P450 2B6(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50505255(BIIB-074 | BIIB074 | CNV-1014802 | CNV1014802 | GS...)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of CYP2B6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544649(CHEMBL4643518)copy SMILEScopy InChI
Affinity DataIC50: 3.16E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544677(CHEMBL4634692)copy SMILEScopy InChI
Affinity DataIC50: 3.16E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544668(CHEMBL4637074)copy SMILEScopy InChI
Affinity DataIC50: 3.16E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544669(CHEMBL4647249)copy SMILEScopy InChI
Affinity DataIC50: 3.98E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544668(CHEMBL4637074)copy SMILEScopy InChI
Affinity DataIC50: 3.98E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544663(CHEMBL4638017)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544679(CHEMBL4633318)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544682(CHEMBL4637843)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544659(CHEMBL4643538)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544663(CHEMBL4638017)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544683(CHEMBL4648908)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544660(CHEMBL4643471)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544653(CHEMBL4646035)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544688(CHEMBL4646990)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544665(CHEMBL4647983)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544680(CHEMBL4638413)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544676(CHEMBL4635121)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544675(CHEMBL4637902)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544674(CHEMBL4645734)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544673(CHEMBL4642930)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50544672(CHEMBL4644773)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
Convergence Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50505255(BIIB-074 | BIIB074 | CNV-1014802 | CNV1014802 | GS...)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+4nMAssay Description:Inhibition of Nav1.3 (unknown origin) expressed in HEK293 cells assessed as inhibition of sodium current incubated for 3 to 3.5 mins by electrophysio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2DHXPubMed
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