TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 0.120nMAssay Description:Displacement of specific [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Displacement of specific [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:Displacement of [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells; ranges from 0.16-0.21More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Displacement of specific [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 0.430nMAssay Description:Displacement of specific [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 0.590nMAssay Description:Displacement of specific [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells; ranges from 0.69-0.92More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of specific [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of specific [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of specific [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of specific [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 1.31nMAssay Description:Displacement of specific [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Displacement of [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells; ranges from 3.4-4.2More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of specific [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 4.40nMAssay Description:Displacement of specific [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 4.63nMAssay Description:Displacement of specific [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 4.80nMAssay Description:Displacement of specific [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 5.48nMAssay Description:Displacement of [3H]-SCH- 58261 from human Adenosine A2A receptor expressed in HEK-293 cells; ranges from 4.95-6.08More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Displacement of specific [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Displacement of [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells; ranges from 48.9-52.4More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Displacement of specific [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Displacement of [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells; ranges from 49-72More data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Displacement of specific [3H]-DPCPX binding at human Adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 75nMAssay Description:Displacement of [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells; ranges from 66-85More data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Displacement of specific [3H]-DPCPX binding at human Adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 86nMAssay Description:Displacement of specific [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Displacement of specific [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Displacement of [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells; ranges from 98-144More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Displacement of [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells; ranges from 98-144More data for this Ligand-Target Pair
Affinity DataKi: 123nMAssay Description:Displacement of specific [3H]-DPCPX binding at human Adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
Affinity DataKi: 139nMAssay Description:Displacement of [3H]-DPCPX from human Adenosine A1 receptor expressed in CHO cells; ranges from 107-181More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 140nMAssay Description:Displacement of [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells; ranges from 129-152More data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Displacement of specific [3H]-DPCPX binding at human Adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Displacement of specific [3H]-DPCPX binding at human Adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
Affinity DataKi: 369nMAssay Description:Displacement of [3H]-DPCPX from human Adenosine A1 receptor expressed in CHO cells; ranges from 324-420More data for this Ligand-Target Pair
Affinity DataKi: 419nMAssay Description:Displacement of specific [3H]-DPCPX binding at human Adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
Affinity DataKi: 432nMAssay Description:Displacement of [3H]-DPCPX binding at human Adenosine A1 receptor expressed in CHO cells; ranges from 363-514More data for this Ligand-Target Pair
Affinity DataKi: 549nMAssay Description:Displacement of specific [3H]-DPCPX binding at human Adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
Affinity DataKi: 558nMAssay Description:Displacement of specific [3H]-DPCPX binding at human Adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
Affinity DataKi: 576nMAssay Description:Displacement of specific [3H]-DPCPX binding at human Adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
Affinity DataKi: 1.03E+3nMAssay Description:Displacement of specific [3H]-DPCPX binding at human Adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
Affinity DataKi: 1.79E+3nMAssay Description:Displacement of [3H]-DPCPX from human Adenosine A1 receptor expressed in CHO cells; ranges from 1460-2201More data for this Ligand-Target Pair
Affinity DataKi: 2.16E+3nMAssay Description:Displacement of specific [3H]-DPCPX binding at human Adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Displacement of [3H]-DPCPX from human Adenosine A1 receptor expressed in CHO cells; ranges from 2153-2891More data for this Ligand-Target Pair
Affinity DataKi: 2.63E+3nMAssay Description:Displacement of specific [3H]-DPCPX binding at human Adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
Affinity DataKi: 3.60E+3nMAssay Description:Displacement of [3H]-DPCPX from human Adenosine A1 receptor expressed in CHO cells; ranges from 3420-3788More data for this Ligand-Target Pair
Affinity DataKi: 4.20E+3nMAssay Description:Displacement of specific [3H]-DPCPX binding at human Adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
Affinity DataKi: 4.49E+3nMAssay Description:Displacement of specific [3H]-DPCPX binding at human Adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
Affinity DataKi: 4.93E+3nMAssay Description:Displacement of specific [3H]-DPCPX binding at human Adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
Affinity DataKi: 4.97E+3nMAssay Description:Displacement of specific [3H]-DPCPX binding at human Adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair