Affinity DataKi: 140nMAssay Description:Inhibition of full length wild type CLK1 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by NanoBRET NanoGlo Substrate additi...More data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Inhibition of full length wild type CLK1 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by NanoBRET NanoGlo Substrate additi...More data for this Ligand-Target Pair
Affinity DataKi: 5.20E+3nMAssay Description:Inhibition of recombinant CLK3 (unknown origin) using Ac-ERMRPRKRQGSVdP(Sox)G-NH2 as substrate after 5 mins by Omnia Kinase AssayMore data for this Ligand-Target Pair
Affinity DataKi: 2.69E+4nMAssay Description:Inhibition of recombinant CLK3 (unknown origin) using Ac-ERMRPRKRQGSVdP(Sox)G-NH2 as substrate after 5 mins by Omnia Kinase AssayMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of human CLK1 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of human CLK4 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of human CLK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of human HIPK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 159nMAssay Description:Inhibition of human HIPK3 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 187nMAssay Description:Inhibition of human HIPK1 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 213nMAssay Description:Inhibition of DYRK1A (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 956nMAssay Description:Inhibition of human DYRK1B by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of human DYRK2 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human CLK3 by radiometric assayMore data for this Ligand-Target Pair
Affinity DataKd: 75nMAssay Description:Inhibition of CLK1 (H148 to I484 residues) (unknown origin) at 15 uM by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Binding affinity to MAP3K19 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Binding affinity to CSNK1E (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Binding affinity to CSNK1D (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Binding affinity to CSNK1G3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Binding affinity to CSNK1G2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Binding affinity to PIM3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Binding affinity to PIM1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 1.00E+3nMAssay Description:Binding affinity to CLK3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: <100nMAssay Description:Binding affinity to CLK4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: <100nMAssay Description:Binding affinity to CLK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: <100nMAssay Description:Binding affinity to CLK1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 7.78E+3nMAssay Description:Inhibition of CLK3 (R134 to T484 residues) (unknown origin) at 15 uM by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Binding affinity to DYRK1A (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Binding affinity to DYRK1B (unknown origin)More data for this Ligand-Target Pair
![](/img/powered_by_small.gif)