Compile Data Set for Download or QSAR
Found 34 Enz. Inhib. hit(s) with all data for entry = 50012851
LigandPNGBDBM50561000(CHEMBL1551597)copy SMILES
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human T type calcium channel Cav3.2 expressed in HEK-293T cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561000(CHEMBL1551597)copy SMILES
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of human N type calcium channel Cav2.2 endogenously expressed in SH-SY5Y cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561005(CHEMBL4741422)copy SMILES
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of human T type calcium channel Cav3.2 expressed in HEK-293T cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50101813(CHEBI:31399 | Cilnidipine)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of human T type calcium channel Cav3.2 expressed in HEK-293T cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50101813(CHEBI:31399 | Cilnidipine)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of human N type calcium channel Cav2.2 endogenously expressed in SH-SY5Y cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561001(CHEMBL4800369)copy SMILES
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of human Cav2.2 expressed in HEK293 cells by whole cell patch clamp electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561010(CHEMBL4794579)copy SMILES
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of human N type calcium channel Cav2.2 endogenously expressed in SH-SY5Y cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561002(CHEMBL4759180)copy SMILES
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of human T type calcium channel Cav3.2 expressed in HEK-293T cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561007(CHEMBL4742798)copy SMILES
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibition of human N type calcium channel Cav2.2 endogenously expressed in SH-SY5Y cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561010(CHEMBL4794579)copy SMILES
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibition of human T type calcium channel Cav3.2 expressed in HEK-293T cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561005(CHEMBL4741422)copy SMILES
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibition of human N type calcium channel Cav2.2 endogenously expressed in SH-SY5Y cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561004(CHEMBL4740547)copy SMILES
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of human T type calcium channel Cav3.2 expressed in HEK-293T cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561007(CHEMBL4742798)copy SMILES
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibition of human T type calcium channel Cav3.2 expressed in HEK-293T cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561006(CHEMBL4764424)copy SMILES
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibition of human T type calcium channel Cav3.2 expressed in HEK-293T cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561006(CHEMBL4764424)copy SMILES
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibition of human N type calcium channel Cav2.2 endogenously expressed in SH-SY5Y cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561014(CHEMBL4794057)copy SMILES
Affinity DataIC50: 7.80E+4nMAssay Description:Inhibition of human N type calcium channel Cav2.2 endogenously expressed in SH-SY5Y cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561009(CHEMBL4781385)copy SMILES
Affinity DataIC50: 7.80E+4nMAssay Description:Inhibition of human N type calcium channel Cav2.2 endogenously expressed in SH-SY5Y cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561014(CHEMBL4794057)copy SMILES
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of human T type calcium channel Cav3.2 expressed in HEK-293T cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561008(CHEMBL4791782)copy SMILES
Affinity DataIC50: 8.70E+4nMAssay Description:Inhibition of human N type calcium channel Cav2.2 endogenously expressed in SH-SY5Y cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561011(CHEMBL4741821)copy SMILES
Affinity DataIC50: 9.80E+4nMAssay Description:Inhibition of human N type calcium channel Cav2.2 endogenously expressed in SH-SY5Y cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561009(CHEMBL4781385)copy SMILES
Affinity DataIC50: 1.02E+5nMAssay Description:Inhibition of human T type calcium channel Cav3.2 expressed in HEK-293T cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561004(CHEMBL4740547)copy SMILES
Affinity DataIC50: 1.02E+5nMAssay Description:Inhibition of human N type calcium channel Cav2.2 endogenously expressed in SH-SY5Y cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561012(CHEMBL4749090)copy SMILES
Affinity DataIC50: 1.07E+5nMAssay Description:Inhibition of human N type calcium channel Cav2.2 endogenously expressed in SH-SY5Y cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561008(CHEMBL4791782)copy SMILES
Affinity DataIC50: 1.08E+5nMAssay Description:Inhibition of human T type calcium channel Cav3.2 expressed in HEK-293T cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561011(CHEMBL4741821)copy SMILES
Affinity DataIC50: 1.10E+5nMAssay Description:Inhibition of human T type calcium channel Cav3.2 expressed in HEK-293T cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561012(CHEMBL4749090)copy SMILES
Affinity DataIC50: 1.13E+5nMAssay Description:Inhibition of human T type calcium channel Cav3.2 expressed in HEK-293T cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561013(CHEMBL4741805)copy SMILES
Affinity DataIC50: 1.29E+5nMAssay Description:Inhibition of human N type calcium channel Cav2.2 endogenously expressed in SH-SY5Y cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561013(CHEMBL4741805)copy SMILES
Affinity DataIC50: 1.33E+5nMAssay Description:Inhibition of human T type calcium channel Cav3.2 expressed in HEK-293T cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561003(CHEMBL4754749)copy SMILES
Affinity DataIC50: 1.64E+5nMAssay Description:Inhibition of human T type calcium channel Cav3.2 expressed in HEK-293T cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561001(CHEMBL4800369)copy SMILES
Affinity DataIC50: 1.85E+5nMAssay Description:Inhibition of human N type calcium channel Cav2.2 endogenously expressed in SH-SY5Y cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561015(CHEMBL4749956)copy SMILES
Affinity DataIC50: 1.93E+5nMAssay Description:Inhibition of human T type calcium channel Cav3.2 expressed in HEK-293T cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561015(CHEMBL4749956)copy SMILES
Affinity DataIC50: 2.59E+5nMAssay Description:Inhibition of human N type calcium channel Cav2.2 endogenously expressed in SH-SY5Y cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561003(CHEMBL4754749)copy SMILES
Affinity DataIC50: 4.04E+5nMAssay Description:Inhibition of human N type calcium channel Cav2.2 endogenously expressed in SH-SY5Y cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed
LigandPNGBDBM50561002(CHEMBL4759180)copy SMILES
Affinity DataIC50: 5.91E+5nMAssay Description:Inhibition of human N type calcium channel Cav2.2 endogenously expressed in SH-SY5Y cells assessed as calcium influx by FRIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B066SPubMed