Found 15 Enz. Inhib. hit(s) with all data for entry = 50012939 
Affinity DataIC50: 20nMAssay Description:Displacement of fluorescent tracer Rap-Gly-BDP from nanoluciferse-tagged human FKBP12 expressed in HEK293T cells incubated for 2 hrs by NanoBRET assa...More data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataIC50: 23nMAssay Description:Displacement of fluorescent probe SLFb-2PEG-TAMRA from N-terminal 6His-SUMO-tagged human full length FKBP12 expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Displacement of fluorescent probe SLFb-2PEG-TAMRA from N-terminal 6His-SUMO-tagged human full length FKBP12 expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Displacement of fluorescent probe SLFb-2PEG-TAMRA from N-terminal 6His-SUMO-tagged human full length FKBP12 expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Displacement of fluorescent probe SLFb-2PEG-TAMRA from N-terminal 6His-SUMO-tagged human full length FKBP12 expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Displacement of fluorescent probe SLFb-2PEG-TAMRA from N-terminal 6His-SUMO-tagged human full length FKBP12 expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Displacement of fluorescent probe SLFb-2PEG-TAMRA from N-terminal 6His-SUMO-tagged human full length FKBP12 expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Displacement of fluorescent probe SLFb-2PEG-TAMRA from N-terminal 6His-SUMO-tagged human full length FKBP12 expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Displacement of fluorescent probe SLFb-2PEG-TAMRA from N-terminal 6His-SUMO-tagged human full length FKBP12 expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
Affinity DataIC50: 132nMAssay Description:Displacement of fluorescent probe SLFb-2PEG-TAMRA from N-terminal 6His-SUMO-tagged human full length FKBP12 expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
Affinity DataIC50: 166nMAssay Description:Displacement of fluorescent probe SLFb-2PEG-TAMRA from N-terminal 6His-SUMO-tagged human full length FKBP12 expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
Affinity DataIC50: 326nMAssay Description:Displacement of fluorescent probe SLFb-2PEG-TAMRA from N-terminal 6His-SUMO-tagged human full length FKBP12 expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
Affinity DataIC50: 423nMAssay Description:Displacement of fluorescent probe SLFb-2PEG-TAMRA from N-terminal 6His-SUMO-tagged human full length FKBP12 expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
Affinity DataIC50: 3.25E+3nMAssay Description:Displacement of fluorescent probe SLFb-2PEG-TAMRA from N-terminal 6His-SUMO-tagged human full length FKBP12 expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
Affinity DataIC50: 3.63E+3nMAssay Description:Displacement of fluorescent probe SLFb-2PEG-TAMRA from N-terminal 6His-SUMO-tagged human full length FKBP12 expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
