Compile Data Set for Download or QSAR
Found 27 Enz. Inhib. hit(s) with all data for entry = 50013414
TargetSerine/threonine-protein kinase D3(Homo sapiens (Human))TBA
LigandPNGBDBM50565693(CHEMBL4515390)copy SMILES
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant FLAG-tagged PKD3 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))TBA
LigandPNGBDBM50565693(CHEMBL4515390)copy SMILES
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))TBA
LigandPNGBDBM50565693(CHEMBL4515390)copy SMILES
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant FLAG-tagged PKD1 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D3(Homo sapiens (Human))TBA
LigandPNGBDBM50565690(CHEMBL4787572)copy SMILES
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant FLAG-tagged PKD3 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))TBA
LigandPNGBDBM50565690(CHEMBL4787572)copy SMILES
Affinity DataIC50: 35nMAssay Description:Inhibition of recombinant FLAG-tagged PKD1 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))TBA
LigandPNGBDBM50565690(CHEMBL4787572)copy SMILES
Affinity DataIC50: 35nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))TBA
LigandPNGBDBM50565692(CHEMBL4790321)copy SMILES
Affinity DataIC50: 43nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D3(Homo sapiens (Human))TBA
LigandPNGBDBM416549(US10307425, Example 15 | US10632122, Example 15)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Inhibition of recombinant FLAG-tagged PKD3 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))TBA
LigandPNGBDBM416549(US10307425, Example 15 | US10632122, Example 15)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))TBA
LigandPNGBDBM50565692(CHEMBL4790321)copy SMILES
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant FLAG-tagged PKD1 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))TBA
LigandPNGBDBM50565691(CHEMBL4776166)copy SMILES
Affinity DataIC50: 55nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))TBA
LigandPNGBDBM50565691(CHEMBL4776166)copy SMILES
Affinity DataIC50: 64nMAssay Description:Inhibition of recombinant FLAG-tagged PKD1 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D3(Homo sapiens (Human))TBA
LigandPNGBDBM50565692(CHEMBL4790321)copy SMILES
Affinity DataIC50: 76nMAssay Description:Inhibition of recombinant FLAG-tagged PKD3 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D3(Homo sapiens (Human))TBA
LigandPNGBDBM50565691(CHEMBL4776166)copy SMILES
Affinity DataIC50: 78nMAssay Description:Inhibition of recombinant FLAG-tagged PKD3 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))TBA
LigandPNGBDBM50565687(CHEMBL4779081)copy SMILES
Affinity DataIC50: 94nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D3(Homo sapiens (Human))TBA
LigandPNGBDBM50565687(CHEMBL4779081)copy SMILES
Affinity DataIC50: 108nMAssay Description:Inhibition of recombinant FLAG-tagged PKD3 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))TBA
LigandPNGBDBM50565687(CHEMBL4779081)copy SMILES
Affinity DataIC50: 108nMAssay Description:Inhibition of recombinant FLAG-tagged PKD1 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))TBA
LigandPNGBDBM416549(US10307425, Example 15 | US10632122, Example 15)copy SMILEScopy InChI
Affinity DataIC50: 183nMAssay Description:Inhibition of recombinant FLAG-tagged PKD1 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))TBA
LigandPNGBDBM50565689(CHEMBL4778331)copy SMILES
Affinity DataIC50: 282nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))TBA
LigandPNGBDBM50565689(CHEMBL4778331)copy SMILES
Affinity DataIC50: 343nMAssay Description:Inhibition of recombinant FLAG-tagged PKD1 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D3(Homo sapiens (Human))TBA
LigandPNGBDBM50565689(CHEMBL4778331)copy SMILES
Affinity DataIC50: 456nMAssay Description:Inhibition of recombinant FLAG-tagged PKD3 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D3(Homo sapiens (Human))TBA
LigandPNGBDBM50298225(CHEMBL2069955 | CHEMBL573578 | NM-PP1 | US10544104...)copy SMILEScopy InChI
Affinity DataIC50: 616nMAssay Description:Inhibition of recombinant FLAG-tagged PKD3 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))TBA
LigandPNGBDBM50298225(CHEMBL2069955 | CHEMBL573578 | NM-PP1 | US10544104...)copy SMILEScopy InChI
Affinity DataIC50: 786nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))TBA
LigandPNGBDBM50298225(CHEMBL2069955 | CHEMBL573578 | NM-PP1 | US10544104...)copy SMILEScopy InChI
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of recombinant FLAG-tagged PKD1 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))TBA
LigandPNGBDBM50565688(CHEMBL4800579)copy SMILES
Affinity DataIC50: 3.29E+3nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))TBA
LigandPNGBDBM50565688(CHEMBL4800579)copy SMILES
Affinity DataIC50: 3.32E+3nMAssay Description:Inhibition of recombinant FLAG-tagged PKD1 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed
TargetSerine/threonine-protein kinase D3(Homo sapiens (Human))TBA
LigandPNGBDBM50565688(CHEMBL4800579)copy SMILES
Affinity DataIC50: 4.06E+3nMAssay Description:Inhibition of recombinant FLAG-tagged PKD3 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5JQGPubMed