Found 34 Enz. Inhib. hit(s) with all data for entry = 50013812 
Affinity DataKi: 25nMAssay Description:Binding affinity to beta2 adrenoceptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity to beta2 adrenoceptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity to beta2 adrenoceptor (unknown origin)More data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataKi: 97nMAssay Description:Binding affinity to beta2 adrenoceptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 0.710nMAssay Description:Agonist activity at human beta2 adrenoceptor expressed in CHO cells assessed as increase in intracellular cAMP level incubated for 1 hr by alphascree...More data for this Ligand-Target Pair
Affinity DataEC50: 2.60nMAssay Description:Agonist activity at human beta2 adrenoceptor expressed in CHO cells assessed as increase in intracellular cAMP level incubated for 1 hr by alphascree...More data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Agonist activity at beta2 adrenoceptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 27nMAssay Description:Agonist activity at beta2 adrenoceptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 0.790nMAssay Description:Agonist activity at beta2 adrenoceptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 0.0200nMAssay Description:Agonist activity at beta2 adrenoceptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 2.90nMAssay Description:Agonist activity at human beta2 adrenoceptor expressed in CHO cells assessed as increase in cAMP level incubated for 30 mins by immunoassayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.40E+3nMAssay Description:Agonist activity at human beta1 adrenoceptor expressed in CHO cells assessed as increase in cAMP level incubated for 30 mins by immunoassayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:Inhibition of 3H]CGP12177 binding to human beta2 adrenoceptor expressed in sf9 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataEC50: 36nMAssay Description:Inhibition of 3H]CGP12177 binding to human beta1 adrenoceptor expressed in sf9 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataEC50: 2.38E+4nMAssay Description:Agonist activity at beta2 adrenoceptor in human A431 cells measured for 24 hrsMore data for this Ligand-Target Pair
Affinity DataEC50: 5.93E+3nMAssay Description:Agonist activity at beta2 adrenoceptor in human A431 cells measured for 24 hrsMore data for this Ligand-Target Pair
Affinity DataEC50: 88nMAssay Description:Agonist activity at beta2 adrenoceptor (unknown origin) expressed in CHO-K1 cells harboring Galpha15 assessed as induction of calcium current by FLIP...More data for this Ligand-Target Pair
Affinity DataEC50: 0.251nMAssay Description:Agonist activity at human beta2 adrenoceptor expressed in HEK293 cells assessed as increase in cAMP accumulation measured after 60 mins by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 195nMAssay Description:Agonist activity at human beta1 adrenoceptor expressed in HEK293 cells assessed as increase in cAMP accumulation measured after 60 mins by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.40E+3nMAssay Description:Agonist activity at beta2 adrenoceptor (unknown origin) expressed in HEK293 cells assessed as increase in isoproterenol-induced cAMP production prein...More data for this Ligand-Target Pair
Affinity DataEC50: 3.20E+3nMAssay Description:Agonist activity at beta2 adrenoceptor (unknown origin) expressed in HEK293 cells co-expressing V2 receptor assessed as induction of beta-arrestin 2 ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+4nMAssay Description:Agonist activity at beta2 adrenoceptor in HEK293 cells co-expressing V2 receptor assessed as increase in cAMP accumulation measured after 30 mins by ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.74E+4nMAssay Description:Agonist activity at beta2 adrenoceptor in HEK293 cells co-expressing V2 receptor assessed as increase in cAMP accumulation measured after 30 mins by ...More data for this Ligand-Target Pair
Affinity DataEC50: 3.55E+4nMAssay Description:Agonist activity at beta2 adrenoceptor in HEK293 cells co-expressing V2 receptor assessed as increase in cAMP accumulation measured after 30 mins by ...More data for this Ligand-Target Pair
Affinity DataEC50: 7.58E+3nMAssay Description:Agonist activity at human beta2 adrenoceptor expressed in CHO cells harboring beta2-beta-arr assessed as induction of beta-arrestin 2 recruitment usi...More data for this Ligand-Target Pair
Affinity DataEC50: 5.01E+3nMAssay Description:Agonist activity at human beta2 adrenoceptor expressed in CHO cells harboring beta2-beta-arr assessed as induction of beta-arrestin 2 recruitment usi...More data for this Ligand-Target Pair
Affinity DataEC50: 6.16E+3nMAssay Description:Agonist activity at human beta2 adrenoceptor expressed in CHO cells harboring beta2-beta-arr assessed as induction of beta-arrestin 2 recruitment usi...More data for this Ligand-Target Pair
Affinity DataEC50: 5.20E+3nMAssay Description:Agonist activity at beta2 adrenoceptor (unknown origin) expressed in sf9 cells assessed as reversal of norepinephrine inhibition of [3H]DHAP binding ...More data for this Ligand-Target Pair
Affinity DataEC50: 3.89E+3nMAssay Description:Agonist activity at beta1 adrenoceptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 251nMAssay Description:Agonist activity at human beta2 adrenoceptor expressed in CHO cells assessed as increase in intracellular cAMP level incubated for 1 hr by alphascree...More data for this Ligand-Target Pair
Affinity DataEC50: 109nMAssay Description:Agonist activity at human beta1 adrenoceptor expressed in CHO cells assessed as increase in intracellular cAMP level incubated for 1 hr by alphascree...More data for this Ligand-Target Pair
Affinity DataEC50: 1.90nMAssay Description:Agonist activity at beta2 adrenoceptor human bronchi assessed as induction of maximum relaxationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.17E+3nMAssay Description:Agonist activity at human beta1 adrenoceptor expressed in CHO cells assessed as increase in intracellular cAMP level incubated for 1 hr by alphascree...More data for this Ligand-Target Pair
Affinity DataEC50: 67nMAssay Description:Agonist activity at human beta1 adrenoceptor expressed in CHO cells assessed as increase in intracellular cAMP level incubated for 1 hr by alphascree...More data for this Ligand-Target Pair
