Compile Data Set for Download or QSAR
Found 42 Enz. Inhib. hit(s) with all data for entry = 50014056
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572196(CHEMBL4879265)copy SMILES
Affinity DataIC50: 4nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572198(CHEMBL4873479)copy SMILES
Affinity DataIC50: 4nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572194(CHEMBL4862136)copy SMILES
Affinity DataIC50: 6nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572195(CHEMBL4868908)copy SMILES
Affinity DataIC50: 7nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572200(CHEMBL4862951)copy SMILES
Affinity DataIC50: 9nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572199(CHEMBL4866999)copy SMILES
Affinity DataIC50: 9nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572201(CHEMBL4864750)copy SMILES
Affinity DataIC50: 9nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572197(CHEMBL4879088)copy SMILES
Affinity DataIC50: 14nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572193(CHEMBL4873185)copy SMILES
Affinity DataIC50: 14nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572192(CHEMBL4858549)copy SMILES
Affinity DataIC50: 26nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572191(CHEMBL4861727)copy SMILES
Affinity DataIC50: 35nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572198(CHEMBL4873479)copy SMILES
Affinity DataIC50: 50nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 assessed as reduction in decatenation using supercoiled pNO1 plasmid DNA as substrate incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572196(CHEMBL4879265)copy SMILES
Affinity DataIC50: 67nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572198(CHEMBL4873479)copy SMILES
Affinity DataIC50: 87nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572196(CHEMBL4879265)copy SMILES
Affinity DataIC50: 90nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 assessed as reduction in decatenation using supercoiled pNO1 plasmid DNA as substrate incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572203(CHEMBL4855172)copy SMILES
Affinity DataIC50: 123nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572201(CHEMBL4864750)copy SMILES
Affinity DataIC50: 126nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572197(CHEMBL4879088)copy SMILES
Affinity DataIC50: 172nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572195(CHEMBL4868908)copy SMILES
Affinity DataIC50: 197nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572197(CHEMBL4879088)copy SMILES
Affinity DataIC50: 215nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 assessed as reduction in decatenation using supercoiled pNO1 plasmid DNA as substrate incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572194(CHEMBL4862136)copy SMILES
Affinity DataIC50: 236nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572195(CHEMBL4868908)copy SMILES
Affinity DataIC50: 241nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 assessed as reduction in decatenation using supercoiled pNO1 plasmid DNA as substrate incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50050549(GSK2140944 | Gepotidacin)copy SMILEScopy InChI
Affinity DataIC50: 244nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30 mins...More data for this Ligand-Target Pair
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572193(CHEMBL4873185)copy SMILES
Affinity DataIC50: 280nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572202(CHEMBL4874688)copy SMILES
Affinity DataIC50: 283nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572200(CHEMBL4862951)copy SMILES
Affinity DataIC50: 326nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572199(CHEMBL4866999)copy SMILES
Affinity DataIC50: 356nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50050549(GSK2140944 | Gepotidacin)copy SMILEScopy InChI
Affinity DataIC50: 374nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30...More data for this Ligand-Target Pair
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572192(CHEMBL4858549)copy SMILES
Affinity DataIC50: 570nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572201(CHEMBL4864750)copy SMILES
Affinity DataIC50: 725nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 assessed as reduction in decatenation using supercoiled pNO1 plasmid DNA as substrate incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572194(CHEMBL4862136)copy SMILES
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 assessed as reduction in decatenation using supercoiled pNO1 plasmid DNA as substrate incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572200(CHEMBL4862951)copy SMILES
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 assessed as reduction in decatenation using supercoiled pNO1 plasmid DNA as substrate incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572191(CHEMBL4861727)copy SMILES
Affinity DataIC50: 1.71E+3nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572199(CHEMBL4866999)copy SMILES
Affinity DataIC50: 1.88E+3nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 assessed as reduction in decatenation using supercoiled pNO1 plasmid DNA as substrate incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572193(CHEMBL4873185)copy SMILES
Affinity DataIC50: 2.13E+3nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 assessed as reduction in decatenation using supercoiled pNO1 plasmid DNA as substrate incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572192(CHEMBL4858549)copy SMILES
Affinity DataIC50: 7.22E+3nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 assessed as reduction in decatenation using supercoiled pNO1 plasmid DNA as substrate incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50050549(GSK2140944 | Gepotidacin)copy SMILEScopy InChI
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 assessed as reduction in decatenation using supercoiled pNO1 plasmid DNA as substrate incubated f...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572203(CHEMBL4855172)copy SMILES
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572191(CHEMBL4861727)copy SMILES
Affinity DataIC50: 1.64E+4nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 assessed as reduction in decatenation using supercoiled pNO1 plasmid DNA as substrate incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572202(CHEMBL4874688)copy SMILES
Affinity DataIC50: 1.98E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as reduction in DNA supercoiling using relaxed pNO1 plasmid DNA as substrate incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572202(CHEMBL4874688)copy SMILES
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 assessed as reduction in decatenation using supercoiled pNO1 plasmid DNA as substrate incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50572203(CHEMBL4855172)copy SMILES
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Staphylococcus aureus topoisomerase 4 assessed as reduction in decatenation using supercoiled pNO1 plasmid DNA as substrate incubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D012JPubMed