Compile Data Set for Download or QSAR
Found 35 Enz. Inhib. hit(s) with all data for entry = 50014619
TargetRibosomal protein S6 kinase alpha-2(Homo sapiens (Human))TBA
LigandPNGBDBM50111385(CHEMBL3604793)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of full length recombinant GST-tagged human RSK3 expressed in insect cell using biotin-labelled AGAGRSRHSSYPAGT-OH as substrate in presenc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))TBA
LigandPNGBDBM50111385(CHEMBL3604793)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of full length recombinant His-tagged human RSK2 expressed in baculovirus expression system using biotin-labelled AGAGRSRHSSYPAGT-OH as su...More data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50111384(CHEMBL3604794)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of full length recombinant His-tagged human RSK1 expressed in baculovirus expression system using biotin-labelled AGAGRSRHSSYPAGT-OH as su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50111385(CHEMBL3604793)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of full length recombinant His-tagged human RSK1 expressed in baculovirus expression system using biotin-labelled AGAGRSRHSSYPAGT-OH as su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))TBA
LigandPNGBDBM50111384(CHEMBL3604794)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of full length recombinant His-tagged human RSK2 expressed in baculovirus expression system using biotin-labelled AGAGRSRHSSYPAGT-OH as su...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578032(CHEMBL4847762)copy SMILES
Affinity DataIC50: 9.5nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM25017(2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimeth...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578046(CHEMBL4846725)copy SMILES
Affinity DataIC50: 12nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578033(CHEMBL4847469)copy SMILES
Affinity DataIC50: 12nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-2(Homo sapiens (Human))TBA
LigandPNGBDBM50111384(CHEMBL3604794)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of full length recombinant GST-tagged human RSK3 expressed in insect cell using biotin-labelled AGAGRSRHSSYPAGT-OH as substrate in presenc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM25017(2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimeth...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of RSK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))TBA
LigandPNGBDBM50248765(1-(4-amino-7-(3-hydroxypropyl)-5-p-tolyl-7H-pyrrol...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of RSK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578034(CHEMBL4870231)copy SMILES
Affinity DataIC50: 15nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578027(CHEMBL4870807)copy SMILES
Affinity DataIC50: 16nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578040(CHEMBL4846978)copy SMILES
Affinity DataIC50: 18nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-2(Homo sapiens (Human))TBA
LigandPNGBDBM25017(2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimeth...)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of RSK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))TBA
LigandPNGBDBM25017(2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimeth...)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of His6-tagged human RSK2 using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK-peptide as substrate in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578031(CHEMBL4845942)copy SMILES
Affinity DataIC50: 25nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578035(CHEMBL4872665)copy SMILES
Affinity DataIC50: 29nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-1(Rattus norvegicus)TBA
LigandPNGBDBM25017(2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimeth...)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of N-terminal HA-tagged rat RSK1 using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK-peptide as substrate in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578043(CHEMBL4852908)copy SMILES
Affinity DataIC50: 33nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578036(CHEMBL4850890)copy SMILES
Affinity DataIC50: 55nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578029(CHEMBL4856762)copy SMILES
Affinity DataIC50: 84nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578024(CHEMBL4869608)copy SMILES
Affinity DataIC50: 117nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578038(CHEMBL4852557)copy SMILES
Affinity DataIC50: 301nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578028(CHEMBL4850184)copy SMILES
Affinity DataIC50: 395nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578039(CHEMBL4874868)copy SMILES
Affinity DataIC50: 410nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578025(CHEMBL4865220)copy SMILES
Affinity DataIC50: 2.12E+3nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578042(CHEMBL4846647)copy SMILES
Affinity DataIC50: 3.59E+3nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578030(CHEMBL4866663)copy SMILES
Affinity DataIC50: 4.73E+3nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578044(CHEMBL4868071)copy SMILES
Affinity DataIC50: 7.34E+3nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578041(CHEMBL4871187)copy SMILES
Affinity DataIC50: 9.74E+3nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578026(CHEMBL4848180)copy SMILES
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578037(CHEMBL4854622)copy SMILES
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50578045(CHEMBL4849875)copy SMILES
Affinity DataIC50: 1.76E+4nMAssay Description:Inhibition of RSK4 (unknown origin) incubated for 40 mins in presence of ATP and lipid substrate by Kinase-Glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD44DCPubMed