Compile Data Set for Download or QSAR
Found 60 Enz. Inhib. hit(s) with all data for entry = 50014689
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146201(6-Phenyl-5-[4-(2-pyrrolidin-1-yl-ethoxy)-phenyl]-5...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146201(6-Phenyl-5-[4-(2-pyrrolidin-1-yl-ethoxy)-phenyl]-5...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146206(2-Benzyl-1-[4-(2-pyrrolidin-1-yl-ethoxy)-phenyl]-1...)copy SMILEScopy InChI
Affinity DataIC50: 4.70nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146200((E)-3-[4-(6-Hydroxy-1-phenyl-3,4-dihydro-1H-isoqui...)copy SMILEScopy InChI
Affinity DataIC50: 4.80nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146223(2-Benzenesulfonyl-1-[4-(2-pyrrolidin-1-yl-ethoxy)-...)copy SMILEScopy InChI
Affinity DataIC50: 5.20nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146216(2-(Naphthalene-1-sulfonyl)-1-[4-(2-pyrrolidin-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 5.60nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146200((E)-3-[4-(6-Hydroxy-1-phenyl-3,4-dihydro-1H-isoqui...)copy SMILEScopy InChI
Affinity DataIC50: 5.90nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146222(1-Benzyl-2-phenyl-1,2,3,4-tetrahydro-isoquinolin-6...)copy SMILEScopy InChI
Affinity DataIC50: 6.70nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146199((E)-3-[4-(6-Hydroxy-1-phenyl-3,4-dihydro-1H-isoqui...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146199((E)-3-[4-(6-Hydroxy-1-phenyl-3,4-dihydro-1H-isoqui...)copy SMILEScopy InChI
Affinity DataIC50: 8.70nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146220(2,2,2-Trifluoro-1-[(R)-6-hydroxy-1-(4-hydroxy-phen...)copy SMILEScopy InChI
Affinity DataIC50: 8.90nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146205(2-Benzo[1,3]dioxol-5-ylmethyl-1-[4-(2-pyrrolidin-1...)copy SMILEScopy InChI
Affinity DataIC50: 9.20nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146207(4-(4-Hydroxy-phenyl)-2-(naphthalene-1-sulfonyl)-1,...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146211(2,2,2-Trifluoro-1-[7-hydroxy-4-(4-hydroxy-phenyl)-...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM20585(2-phenyl-1-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-1...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146198(2-Benzyl-4-(4-hydroxy-phenyl)-1,2,3,4-tetrahydro-i...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146223(2-Benzenesulfonyl-1-[4-(2-pyrrolidin-1-yl-ethoxy)-...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146198(2-Benzyl-4-(4-hydroxy-phenyl)-1,2,3,4-tetrahydro-i...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146216(2-(Naphthalene-1-sulfonyl)-1-[4-(2-pyrrolidin-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146204(1-[1-(4-Bromo-phenyl)-6-hydroxy-3,4-dihydro-1H-iso...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM20585(2-phenyl-1-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-1...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146208(1-[4-(2-Pyrrolidin-1-yl-ethoxy)-phenyl]-2-(toluene...)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146221(2-Phenyl-1-thiophen-2-yl-1,2,3,4-tetrahydro-isoqui...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146215(2,2,2-Trifluoro-1-(6-hydroxy-1-phenyl-3,4-dihydro-...)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146213(CHEMBL93207 | [7-Hydroxy-4-(4-hydroxy-phenyl)-3,4-...)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146207(4-(4-Hydroxy-phenyl)-2-(naphthalene-1-sulfonyl)-1,...)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146202(2,2,2-Trifluoro-1-{6-hydroxy-1-[4-(2-pyrrolidin-1-...)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146226(2-(4-Propyl-benzenesulfonyl)-1-[4-(2-pyrrolidin-1-...)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146209(1-Cyclohexyl-2-phenyl-1,2,3,4-tetrahydro-isoquinol...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146224(1,2-Diphenyl-1,2,3,4-tetrahydro-isoquinolin-6-ol |...)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146206(2-Benzyl-1-[4-(2-pyrrolidin-1-yl-ethoxy)-phenyl]-1...)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146225(2-Benzenesulfonyl-4-(4-hydroxy-phenyl)-1,2,3,4-tet...)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146212(1-Isopropyl-2-phenyl-1,2,3,4-tetrahydro-isoquinoli...)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146219(6-Hydroxy-1-[4-(2-pyrrolidin-1-yl-ethoxy)-phenyl]-...)copy SMILEScopy InChI
Affinity DataIC50: 44nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146224(1,2-Diphenyl-1,2,3,4-tetrahydro-isoquinolin-6-ol |...)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146221(2-Phenyl-1-thiophen-2-yl-1,2,3,4-tetrahydro-isoqui...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146218(1-Cyclohexylmethyl-2-phenyl-1,2,3,4-tetrahydro-iso...)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146220(2,2,2-Trifluoro-1-[(R)-6-hydroxy-1-(4-hydroxy-phen...)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146214(2,2,2-Trifluoro-1-(6-hydroxy-1-thiophen-2-yl-3,4-d...)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146222(1-Benzyl-2-phenyl-1,2,3,4-tetrahydro-isoquinolin-6...)copy SMILEScopy InChI
Affinity DataIC50: 66nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146208(1-[4-(2-Pyrrolidin-1-yl-ethoxy)-phenyl]-2-(toluene...)copy SMILEScopy InChI
Affinity DataIC50: 71nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146202(2,2,2-Trifluoro-1-{6-hydroxy-1-[4-(2-pyrrolidin-1-...)copy SMILEScopy InChI
Affinity DataIC50: 93nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146209(1-Cyclohexyl-2-phenyl-1,2,3,4-tetrahydro-isoquinol...)copy SMILEScopy InChI
Affinity DataIC50: 99nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146217(2-(Naphthalene-2-sulfonyl)-1-[4-(2-pyrrolidin-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 112nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146225(2-Benzenesulfonyl-4-(4-hydroxy-phenyl)-1,2,3,4-tet...)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146211(2,2,2-Trifluoro-1-[7-hydroxy-4-(4-hydroxy-phenyl)-...)copy SMILEScopy InChI
Affinity DataIC50: 123nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146226(2-(4-Propyl-benzenesulfonyl)-1-[4-(2-pyrrolidin-1-...)copy SMILEScopy InChI
Affinity DataIC50: 133nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146213(CHEMBL93207 | [7-Hydroxy-4-(4-hydroxy-phenyl)-3,4-...)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146204(1-[1-(4-Bromo-phenyl)-6-hydroxy-3,4-dihydro-1H-iso...)copy SMILEScopy InChI
Affinity DataIC50: 165nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor alpha expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50146212(1-Isopropyl-2-phenyl-1,2,3,4-tetrahydro-isoquinoli...)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:In vitro concentration required to inhibit [3H]-estradiol binding to human estrogen receptor beta expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67GBKPubMed
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