Compile Data Set for Download or QSAR
Found 41 Enz. Inhib. hit(s) with all data for entry = 50014698
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579208(CHEMBL4867107)copy SMILES
Affinity DataIC50: 2nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579222(CHEMBL4861383)copy SMILES
Affinity DataIC50: 2.30nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518531(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 2.40nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518527(2-Alyl-6-((2′,3′-dihydro-1′H-spi...)copy SMILES
Affinity DataIC50: 2.40nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518526(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 2.40nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518538(2-Allyl-6-((2-(2-hydroxyethyl)-1,2,3,4-tetrahydroi...)copy SMILES
Affinity DataIC50: 2.5nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579228(CHEMBL4867211)copy SMILES
Affinity DataIC50: 2.5nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579214(CHEMBL4856035)copy SMILES
Affinity DataIC50: 2.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579225(CHEMBL4874546)copy SMILES
Affinity DataIC50: 2.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518540(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 2.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518530(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 2.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579218(CHEMBL4876612)copy SMILES
Affinity DataIC50: 2.90nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579223(CHEMBL4853285)copy SMILES
Affinity DataIC50: 3.10nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579224(CHEMBL4861351)copy SMILES
Affinity DataIC50: 3.20nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579227(CHEMBL4847705)copy SMILES
Affinity DataIC50: 3.20nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579221(CHEMBL4866800)copy SMILES
Affinity DataIC50: 3.20nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579216(CHEMBL4865963)copy SMILES
Affinity DataIC50: 3.30nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579213(CHEMBL4853973)copy SMILES
Affinity DataIC50: 3.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579220(CHEMBL4868683)copy SMILES
Affinity DataIC50: 3.70nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579219(CHEMBL4857841)copy SMILES
Affinity DataIC50: 3.70nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579217(CHEMBL4871593)copy SMILES
Affinity DataIC50: 3.90nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579215(CHEMBL4861168)copy SMILES
Affinity DataIC50: 4.60nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579211(CHEMBL4871803)copy SMILES
Affinity DataIC50: 4.80nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579212(CHEMBL4879157)copy SMILES
Affinity DataIC50: 5.20nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579210(CHEMBL4853185)copy SMILES
Affinity DataIC50: 5.70nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579210(CHEMBL4853185)copy SMILES
Affinity DataIC50: 5.70nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579209(CHEMBL4874090)copy SMILES
Affinity DataIC50: 6.40nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579226(CHEMBL4856253)copy SMILES
Affinity DataIC50: 12nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579229(CHEMBL4863657)copy SMILES
Affinity DataIC50: 22nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetSerine/threonine-protein kinase PLK2(Homo sapiens (Human))TBA
LigandPNGBDBM50579217(CHEMBL4871593)copy SMILES
Affinity DataIC50: 40nMAssay Description:Inhibition of PLK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
LigandPNGBDBM50579217(CHEMBL4871593)copy SMILES
Affinity DataIC50: 59nMAssay Description:Inhibition of YSK4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50579217(CHEMBL4871593)copy SMILES
Affinity DataIC50: 60nMAssay Description:Inhibition of EGFR d747-749/A750P mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579231(CHEMBL4847051)copy SMILES
Affinity DataIC50: 64nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetSerine/threonine-protein kinase PLK3(Homo sapiens (Human))TBA
LigandPNGBDBM50579217(CHEMBL4871593)copy SMILES
Affinity DataIC50: 70nMAssay Description:Inhibition of PLK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50579230(CHEMBL4877772)copy SMILES
Affinity DataIC50: 100nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50579217(CHEMBL4871593)copy SMILES
Affinity DataIC50: 227nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50579208(CHEMBL4867107)copy SMILES
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50579217(CHEMBL4871593)copy SMILES
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed
LigandPNGBDBM50579217(CHEMBL4871593)copy SMILES
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8JQMPubMed