Compile Data Set for Download or QSAR
Found 29 Enz. Inhib. hit(s) with all data for entry = 50014715
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50361146(CHEMBL1933775)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579405(CHEMBL4874810)copy SMILES
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579402(CHEMBL4847015)copy SMILES
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579406(CHEMBL4848475)copy SMILES
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579398(CHEMBL4852369)copy SMILES
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50361146(CHEMBL1933775)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579390(CHEMBL1571747)copy SMILES
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579397(CHEMBL4866724)copy SMILES
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579412(CHEMBL4872349)copy SMILES
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579401(CHEMBL4856042)copy SMILES
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579400(CHEMBL4875646)copy SMILES
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579403(CHEMBL3114983)copy SMILES
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579404(CHEMBL4877978)copy SMILES
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579408(CHEMBL4865114)copy SMILES
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50361145(CHEMBL1933774)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579396(CHEMBL4862624)copy SMILES
Affinity DataIC50: 4.10E+4nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579409(CHEMBL4847682)copy SMILES
Affinity DataIC50: 5.70E+4nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579411(CHEMBL4873031)copy SMILES
Affinity DataIC50: 6.80E+4nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579399(CHEMBL4854761)copy SMILES
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579392(CHEMBL4861268)copy SMILES
Affinity DataIC50: 7.20E+4nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50361140(CHEMBL1933615)copy SMILEScopy InChI
Affinity DataIC50: 7.40E+4nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50447934(CHEMBL3114982)copy SMILEScopy InChI
Affinity DataIC50: 7.60E+4nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579393(CHEMBL4851617)copy SMILES
Affinity DataIC50: 1.06E+5nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579410(CHEMBL4854213)copy SMILES
Affinity DataIC50: 1.91E+5nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579407(CHEMBL4875827)copy SMILES
Affinity DataIC50: 1.99E+5nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579394(CHEMBL4852545)copy SMILES
Affinity DataIC50: 2.74E+5nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579391(CHEMBL4857264)copy SMILES
Affinity DataIC50: 3.47E+5nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579395(CHEMBL4870552)copy SMILES
Affinity DataIC50: 4.37E+5nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed
TargetLysine-specific demethylase 4E(Homo sapiens (Human))TBA
LigandPNGBDBM50579390(CHEMBL1571747)copy SMILES
Affinity DataIC50: 5.81E+5nMAssay Description:Inhibition of N-terminal His6-tagged KDM4E (1 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)-R3 preincubated for 10 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28D0130PubMed