Compile Data Set for Download or QSAR
Found 14 Enz. Inhib. hit(s) with all data for entry = 50014736
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579614(CHEMBL4871970)copy SMILES
Affinity DataIC50: 1.60nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579610(CHEMBL4873520)copy SMILES
Affinity DataIC50: 2.20nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579616(CHEMBL4845730)copy SMILES
Affinity DataIC50: 3.20nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579611(CHEMBL4871097)copy SMILES
Affinity DataIC50: 3.90nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579615(CHEMBL4865209)copy SMILES
Affinity DataIC50: 5nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50577458(CHEMBL4858437)copy SMILES
Affinity DataIC50: 16nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579613(CHEMBL4850423)copy SMILES
Affinity DataIC50: 25nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579609(CHEMBL4872874)copy SMILES
Affinity DataIC50: 46nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579618(CHEMBL4871090)copy SMILES
Affinity DataIC50: 67nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579612(CHEMBL4847500)copy SMILES
Affinity DataIC50: 104nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579608(CHEMBL4849969)copy SMILES
Affinity DataIC50: 370nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579617(CHEMBL4863411)copy SMILES
Affinity DataIC50: 5.74E+3nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579607(CHEMBL4865167)copy SMILES
Affinity DataIC50: 8.78E+3nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579606(CHEMBL4851004)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed