Compile Data Set for Download or QSAR
Found 48 Enz. Inhib. hit(s) with all data for entry = 50015293
LigandPNGBDBM50585046(CHEMBL5086263)copy SMILES
Affinity DataIC50: 3nMAssay Description:Inhibition of DYRK1A (unknown origin) at 1 uM by kinomescan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585046(CHEMBL5086263)copy SMILES
Affinity DataIC50: 3nMAssay Description:Inhibition of DYRK1A (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585046(CHEMBL5086263)copy SMILES
Affinity DataIC50: 5nMAssay Description:Inhibition of DYRK1B (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585046(CHEMBL5086263)copy SMILES
Affinity DataIC50: 5nMAssay Description:Inhibition of DYRK1B (unknown origin) at 1 uM by kinomescan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of DYRK1A (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
LigandPNGBDBM50585053(CHEMBL5089965)copy SMILES
Affinity DataIC50: 12nMAssay Description:Inhibition of DYRK1A (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585047(CHEMBL5075335)copy SMILES
Affinity DataIC50: 13nMAssay Description:Inhibition of DYRK1A (unknown origin) at 1 uM by kinomescan methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585045(CHEMBL5093741)copy SMILES
Affinity DataIC50: 13nMAssay Description:Inhibition of DYRK1A (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585053(CHEMBL5089965)copy SMILES
Affinity DataIC50: 18nMAssay Description:Inhibition of DYRK1B (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585047(CHEMBL5075335)copy SMILES
Affinity DataIC50: 19nMAssay Description:Inhibition of DYRK1B (unknown origin) at 1 uM by kinomescan methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585045(CHEMBL5093741)copy SMILES
Affinity DataIC50: 19nMAssay Description:Inhibition of DYRK1B (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
TargetRibosomal protein S6 kinase alpha-6(Homo sapiens (Human))TBA
LigandPNGBDBM50585046(CHEMBL5086263)copy SMILES
Affinity DataIC50: 37nMAssay Description:Inhibition of RSK4 (unknown origin) at 1 uM by kinome scan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585049(CHEMBL5075321)copy SMILES
Affinity DataIC50: 44nMAssay Description:Inhibition of DYRK1A (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585049(CHEMBL5075321)copy SMILES
Affinity DataIC50: 55nMAssay Description:Inhibition of DYRK1B (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
TargetRibosomal protein S6 kinase alpha-2(Homo sapiens (Human))TBA
LigandPNGBDBM50585046(CHEMBL5086263)copy SMILES
Affinity DataIC50: 61nMAssay Description:Inhibition of RSK3 (unknown origin) in human CAL-27 cells measured after 6 hrs by select screen kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585047(CHEMBL5075335)copy SMILES
Affinity DataIC50: 70nMAssay Description:Inhibition of DYRK1B (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Inhibition of DYRK1A (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))TBA
LigandPNGBDBM50585046(CHEMBL5086263)copy SMILES
Affinity DataIC50: 80nMAssay Description:Inhibition of RSK2 (unknown origin) in human CAL-27 cells measured after 6 hrs by select screen kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50585046(CHEMBL5086263)copy SMILES
Affinity DataIC50: 82nMAssay Description:Inhibition of RSK1 (unknown origin) in human CAL-27 cells measured after 6 hrs by select screen kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585050(CHEMBL5081601)copy SMILES
Affinity DataIC50: 86nMAssay Description:Inhibition of DYRK1A (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
TargetTRAF2 and NCK-interacting protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50585045(CHEMBL5093741)copy SMILES
Affinity DataIC50: 87nMAssay Description:Inhibition of TNIK (unknown origin) at 1 uM by kinome scan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50585046(CHEMBL5086263)copy SMILES
Affinity DataIC50: 90nMAssay Description:Inhibition of FAK (unknown origin) in human CAL-27 cells measured after 6 hrs by select screen kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
TargetMisshapen-like kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50585046(CHEMBL5086263)copy SMILES
Affinity DataIC50: 115nMAssay Description:Inhibition of MINK1 (unknown origin) at 1 uM by kinome scan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585046(CHEMBL5086263)copy SMILES
Affinity DataIC50: 132nMAssay Description:Inhibition of MEK4 (unknown origin) at 1 uM by kinome scan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585050(CHEMBL5081601)copy SMILES
Affinity DataIC50: 146nMAssay Description:Inhibition of DYRK1B (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585048(CHEMBL5079894)copy SMILES
Affinity DataIC50: 150nMAssay Description:Inhibition of DYRK1B (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585047(CHEMBL5075335)copy SMILES
Affinity DataIC50: 158nMAssay Description:Inhibition of DYRK1A (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585045(CHEMBL5093741)copy SMILES
Affinity DataIC50: 173nMAssay Description:Inhibition of MEK4 (unknown origin) at 1 uM by kinome scan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))TBA
LigandPNGBDBM50585046(CHEMBL5086263)copy SMILES
Affinity DataIC50: 182nMAssay Description:Inhibition of RSK2 (unknown origin) at 1 uM by kinome scan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585048(CHEMBL5079894)copy SMILES
Affinity DataIC50: 200nMAssay Description:Inhibition of DYRK1A (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
TargetFocal adhesion kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50585046(CHEMBL5086263)copy SMILES
Affinity DataIC50: 210nMAssay Description:Inhibition of FAK (unknown origin) at 1 uM by kinome scan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))TBA
LigandPNGBDBM50585045(CHEMBL5093741)copy SMILES
Affinity DataIC50: 212nMAssay Description:Inhibition of SGK (unknown origin) at 1 uM by kinome scan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585051(CHEMBL5086482)copy SMILES
Affinity DataIC50: 327nMAssay Description:Inhibition of DYRK1A (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50391956(CHEMBL2152265)copy SMILEScopy InChI
Affinity DataIC50: 329nMAssay Description:Inhibition of DYRK1A (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
TargetMyosin light chain kinase, smooth muscle(Homo sapiens (Human))TBA
LigandPNGBDBM50585045(CHEMBL5093741)copy SMILES
Affinity DataIC50: 334nMAssay Description:Inhibition of MYLK (unknown origin) at 1 uM by kinome scan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50585045(CHEMBL5093741)copy SMILES
Affinity DataIC50: 354nMAssay Description:Inhibition of FLT3 (unknown origin) at 1 uM by kinome scan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50585045(CHEMBL5093741)copy SMILES
Affinity DataIC50: 477nMAssay Description:Inhibition of TRKA (unknown origin) at 1 uM by kinome scan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585051(CHEMBL5086482)copy SMILES
Affinity DataIC50: 533nMAssay Description:Inhibition of DYRK1B (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585052(CHEMBL5089643)copy SMILES
Affinity DataIC50: 582nMAssay Description:Inhibition of DYRK1A (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))TBA
LigandPNGBDBM50585046(CHEMBL5086263)copy SMILES
Affinity DataIC50: 690nMAssay Description:Inhibition of SGK (unknown origin) at 1 uM by kinome scan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585045(CHEMBL5093741)copy SMILES
Affinity DataIC50: 830nMAssay Description:Inhibition of CAMK1B (unknown origin) at 1 uM by kinome scan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585052(CHEMBL5089643)copy SMILES
Affinity DataIC50: 929nMAssay Description:Inhibition of DYRK1B (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50585046(CHEMBL5086263)copy SMILES
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of JNK2 (unknown origin) in human CAL-27 cells measured after 6 hrs by select screen kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))TBA
LigandPNGBDBM50585046(CHEMBL5086263)copy SMILES
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of JNK1 (unknown origin) in human CAL-27 cells measured after 6 hrs by select screen kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585046(CHEMBL5086263)copy SMILES
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of YSK4 (unknown origin) at 1 uM by kinome scan methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585054(CHEMBL5088208)copy SMILES
Affinity DataIC50: 3.05E+3nMAssay Description:Inhibition of DYRK1B (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
LigandPNGBDBM50585054(CHEMBL5088208)copy SMILES
Affinity DataIC50: 3.05E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) measured after 6 hrs in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))TBA
LigandPNGBDBM50585046(CHEMBL5086263)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of JNK3 (unknown origin) in human CAL-27 cells measured after 6 hrs by select screen kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183BDBPubMed