Compile Data Set for Download or QSAR
Found 79 Enz. Inhib. hit(s) with all data for entry = 50016073
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)copy SMILEScopy InChI
Affinity DataKi:  0.650nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0MHVPubMed
TargetAurora kinase B(Homo sapiens (Human))TBA
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)copy SMILEScopy InChI
Affinity DataKi:  3.40nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0MHVPubMed
TargetAurora kinase C(Homo sapiens (Human))TBA
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)copy SMILEScopy InChI
Affinity DataKi:  4.60nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0MHVPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))TBA
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)copy SMILEScopy InChI
Affinity DataKi:  7.70nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0MHVPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))TBA
LigandPNGBDBM50591934(CHEMBL5209160)copy SMILES
Affinity DataIC50: 0.100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0MHVPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))TBA
LigandPNGBDBM50591949(CHEMBL5185001)copy SMILES
Affinity DataIC50: 0.200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0MHVPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))TBA
LigandPNGBDBM50591932(CHEMBL5171469)copy SMILES
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0MHVPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))TBA
LigandPNGBDBM50591954(CHEMBL5183346)copy SMILES
Affinity DataIC50: 0.700nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0MHVPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))TBA
LigandPNGBDBM50591926(CHEMBL5171233)copy SMILES
Affinity DataIC50: 0.700nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0MHVPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))TBA
LigandPNGBDBM50591931(CHEMBL5200865)copy SMILES
Affinity DataIC50: 0.800nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0MHVPubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))TBA
LigandPNGBDBM50073587(CHEMBL3408947 | US10358436, Example A185 | US20230...)copy SMILES
Affinity DataIC50: 4.90nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0MHVPubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))TBA
LigandPNGBDBM50591962(CHEMBL5175418)copy SMILES
Affinity DataIC50: 5.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0MHVPubMed
TargetSerine/threonine-protein kinase Chk2(Homo sapiens (Human))TBA
LigandPNGBDBM50426474(CHEMBL1980391)copy SMILEScopy InChI
Affinity DataIC50: 24nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0MHVPubMed
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50426474(CHEMBL1980391)copy SMILEScopy InChI
Affinity DataIC50: 58nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0MHVPubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))TBA
LigandPNGBDBM50591934(CHEMBL5209160)copy SMILES
Affinity DataIC50: 96nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0MHVPubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))TBA
LigandPNGBDBM50591948(CHEMBL5188129)copy SMILES
Affinity DataIC50: 231nMMore data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VX0MHVPubMed
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