Compile Data Set for Download or QSAR
Found 170 Enz. Inhib. hit(s) with all data for entry = 50016297
LigandPNGBDBM431646(5-[[(2S)-1-(3-Oxo-3-[4-[5-(trifluoromethyl)pyrimid...)copy SMILES
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP14(Homo sapiens (Human))TBA
LigandPNGBDBM434315(US10562891, Example 235 | US11008308, Example 235)copy SMILES
LigandPNGBDBM50594012(CHEMBL5191676)copy SMILES
Affinity DataIC50: 14nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50594006(CHEMBL5192839)copy SMILES
Affinity DataIC50: 130nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50594006(CHEMBL5192839)copy SMILES
Affinity DataIC50: 135nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50594005(CHEMBL5181947)copy SMILES
Affinity DataIC50: 135nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50594005(CHEMBL5181947)copy SMILES
Affinity DataIC50: 140nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50594010(CHEMBL5200358)copy SMILES
Affinity DataIC50: 150nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50594010(CHEMBL5200358)copy SMILES
Affinity DataIC50: 151nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50594007(CHEMBL5187187)copy SMILES
Affinity DataIC50: 155nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50594011(CHEMBL5200521)copy SMILES
Affinity DataIC50: 158nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50594007(CHEMBL5187187)copy SMILES
Affinity DataIC50: 160nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50594011(CHEMBL5200521)copy SMILES
Affinity DataIC50: 160nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))TBA
LigandPNGBDBM50594013(CHEMBL5195249)copy SMILES
Affinity DataIC50: 200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50593992(CHEMBL5186967)copy SMILES
Affinity DataIC50: 288nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50593992(CHEMBL5186967)copy SMILES
Affinity DataIC50: 290nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50594008(CHEMBL5181107)copy SMILES
Affinity DataIC50: 309nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50594008(CHEMBL5181107)copy SMILES
Affinity DataIC50: 310nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))TBA
LigandPNGBDBM50594006(CHEMBL5192839)copy SMILES
Affinity DataIC50: 320nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))TBA
LigandPNGBDBM50594006(CHEMBL5192839)copy SMILES
Affinity DataIC50: 324nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM199181(4-[(4-Carbamoylcyclohexyl)oxy]cyclohexane-1-carbox...)copy SMILEScopy InChI
Affinity DataIC50: 330nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))TBA
LigandPNGBDBM50594010(CHEMBL5200358)copy SMILES
Affinity DataIC50: 363nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))TBA
LigandPNGBDBM50594007(CHEMBL5187187)copy SMILES
Affinity DataIC50: 370nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))TBA
LigandPNGBDBM50594010(CHEMBL5200358)copy SMILES
Affinity DataIC50: 370nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))TBA
LigandPNGBDBM50594007(CHEMBL5187187)copy SMILES
Affinity DataIC50: 370nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))TBA
LigandPNGBDBM50594011(CHEMBL5200521)copy SMILES
Affinity DataIC50: 398nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))TBA
LigandPNGBDBM50594005(CHEMBL5181947)copy SMILES
Affinity DataIC50: 398nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))TBA
LigandPNGBDBM50594005(CHEMBL5181947)copy SMILES
Affinity DataIC50: 400nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))TBA
LigandPNGBDBM50594011(CHEMBL5200521)copy SMILES
Affinity DataIC50: 400nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))TBA
LigandPNGBDBM50594001(CHEMBL5186481)copy SMILES
Affinity DataIC50: 589nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50593991(CHEMBL5206305)copy SMILES
Affinity DataIC50: 589nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50593991(CHEMBL5206305)copy SMILES
Affinity DataIC50: 590nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50593993(CHEMBL5198692)copy SMILES
Affinity DataIC50: 600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))TBA
LigandPNGBDBM50594001(CHEMBL5186481)copy SMILES
Affinity DataIC50: 600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50593993(CHEMBL5198692)copy SMILES
Affinity DataIC50: 603nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50594000(CHEMBL5183715)copy SMILES
Affinity DataIC50: 617nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50594000(CHEMBL5183715)copy SMILES
Affinity DataIC50: 620nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50593999(CHEMBL5198984)copy SMILES
Affinity DataIC50: 955nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50593999(CHEMBL5198984)copy SMILES
Affinity DataIC50: 960nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50594009(CHEMBL5171357)copy SMILES
Affinity DataIC50: 1.15E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50594009(CHEMBL5171357)copy SMILES
Affinity DataIC50: 1.20E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))TBA
LigandPNGBDBM50594008(CHEMBL5181107)copy SMILES
Affinity DataIC50: 1.20E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))TBA
LigandPNGBDBM50594008(CHEMBL5181107)copy SMILES
Affinity DataIC50: 1.20E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))TBA
LigandPNGBDBM50594009(CHEMBL5171357)copy SMILES
Affinity DataIC50: 1.30E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP15(Homo sapiens (Human))TBA
LigandPNGBDBM50594009(CHEMBL5171357)copy SMILES
Affinity DataIC50: 1.35E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM199181(4-[(4-Carbamoylcyclohexyl)oxy]cyclohexane-1-carbox...)copy SMILEScopy InChI
Affinity DataIC50: 1.35E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50594001(CHEMBL5186481)copy SMILES
Affinity DataIC50: 1.50E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50593994(CHEMBL5185078)copy SMILES
Affinity DataIC50: 1.60E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50593990(CHEMBL5178227)copy SMILES
Affinity DataIC50: 1.70E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP10(Homo sapiens (Human))TBA
LigandPNGBDBM50593990(CHEMBL5178227)copy SMILES
Affinity DataIC50: 1.74E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
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