Compile Data Set for Download or QSAR
Found 28 Enz. Inhib. hit(s) with all data for entry = 50016850
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174413(2-(2-Diethylamino-ethyl)-9-hydroxy-5,11-dimethyl-6...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004235((NMHE)9-Hydroxy-2,5,11-trimethyl-6H-pyrido[4,3-b]c...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004227(5,11-Dimethyl-6H-pyrido[4,3-b]carbazol-9-ol | 5,11...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibitory activity against Fibroblast growth factor receptor 3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004227(5,11-Dimethyl-6H-pyrido[4,3-b]carbazol-9-ol | 5,11...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004227(5,11-Dimethyl-6H-pyrido[4,3-b]carbazol-9-ol | 5,11...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004235((NMHE)9-Hydroxy-2,5,11-trimethyl-6H-pyrido[4,3-b]c...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174413(2-(2-Diethylamino-ethyl)-9-hydroxy-5,11-dimethyl-6...)copy SMILEScopy InChI
Affinity DataIC50: 450nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004235((NMHE)9-Hydroxy-2,5,11-trimethyl-6H-pyrido[4,3-b]c...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibitory activity against Fibroblast growth factor receptor 3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174412(9-Methoxy-5,11-dimethyl-6H-pyrido[4,3-b]carbazole ...)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004227(5,11-Dimethyl-6H-pyrido[4,3-b]carbazol-9-ol | 5,11...)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibitory activity against Platelet-derived growth factor receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004235((NMHE)9-Hydroxy-2,5,11-trimethyl-6H-pyrido[4,3-b]c...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against Platelet-derived growth factor receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174412(9-Methoxy-5,11-dimethyl-6H-pyrido[4,3-b]carbazole ...)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174410(1-(3-Diethylamino-propylamino)-5,11-dimethyl-6H-py...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174410(1-(3-Diethylamino-propylamino)-5,11-dimethyl-6H-py...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174408(1-(3-Diethylamino-propylamino)-5,6,11-trimethyl-6H...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory activity against Fibroblast growth factor receptor 3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174411(CHEMBL197610 | N,N-Diethyl-N'-(10-methyl-11H-pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174408(1-(3-Diethylamino-propylamino)-5,6,11-trimethyl-6H...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against Platelet-derived growth factor receptor alphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174407(CHEMBL279472 | N,N-Diethyl-N'-(9-methoxy-5-methyl-...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174411(CHEMBL197610 | N,N-Diethyl-N'-(10-methyl-11H-pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174407(CHEMBL279472 | N,N-Diethyl-N'-(9-methoxy-5-methyl-...)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174408(1-(3-Diethylamino-propylamino)-5,6,11-trimethyl-6H...)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174408(1-(3-Diethylamino-propylamino)-5,6,11-trimethyl-6H...)copy SMILEScopy InChI
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004233(5,11-dimethyl-2H-pyrido[4,3-b]carbazole | CHEMBL12...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174409(9-Bromo-5,11-dimethyl-6H-pyrido[4,3-b]carbazole | ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50004233(5,11-dimethyl-2H-pyrido[4,3-b]carbazole | CHEMBL12...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM50174409(9-Bromo-5,11-dimethyl-6H-pyrido[4,3-b]carbazole | ...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against c-Kit wild type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
CNRS UMR-8113

Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against c-Kit D816V type expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27TTRPubMed