Affinity DataKi: 6.80nMAssay Description:Tested for its antagonist activity against mu receptor using DAMGO as radioligand in isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataKi: 7.70nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
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In DepthDetails
Affinity DataKi: 25nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails
Affinity DataKi: 109nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
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In DepthDetails
Affinity DataKi: 620nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails
Affinity DataKi: 620nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
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UniProtKB/SwissProt
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In DepthDetails
Affinity DataKi: 916nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
Affinity DataKi: 5.50E+3nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
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UniProtKB/SwissProt
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In DepthDetails
Affinity DataKi: 1.10E+4nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Affinity DataKi: 3.60E+4nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataKi: 5.40E+4nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
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UniProtKB/SwissProt
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In DepthDetails
Affinity DataKi: 5.40E+4nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
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UniProtKB/SwissProt
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In DepthDetails
Affinity DataKi: 6.90E+4nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
Affinity DataKi: 7.00E+4nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.210nMAssay Description:Antagonist activity at NK-2 tachykinin receptors in rabbit pulmonary arteryMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 0.210nMAssay Description:Tested for inhibitory activity against (DPDE)delta receptor in mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Tested for its antagonist activity against mu receptor using DAMGO as radioligand in isolated guinea pig ileumMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
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In DepthDetails
Affinity DataIC50: 17nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]; inactive up to a co...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 17nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
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UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
In DepthDetails
Affinity DataIC50: 19nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
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UniProtKB/SwissProt
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In DepthDetails
Affinity DataIC50: 25nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 33nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 41nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
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UniProtKB/SwissProt
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In DepthDetails
Affinity DataIC50: 110nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 145nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 550nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 3.00E+3nMAssay Description:Tested for its antagonist activity against kappa receptor using U-69,593 as radioligand in isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 3.70E+3nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]; inactive up to a co...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at NK-2 tachykinin receptors in rabbit pulmonary arteryMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
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UniProtKB/SwissProt
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In DepthDetails
Affinity DataKd: 216nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
In DepthDetails
Affinity DataKd: 27nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]; inactive up to a co...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataEC50: 2.60E+4nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
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UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
In DepthDetails
Affinity DataEC50: 2.30E+3nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails
Affinity DataKd: 210nMAssay Description:Tested for its antagonist activity against kappa receptor using U-69,593 as radioligand in isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataKd: 43nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails
Affinity DataKd: 25nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails
Affinity DataKd: <100nMAssay Description:Tested for antagonist activity at NK-2 tachykinin receptors in hamster tracheaMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataKd: 149nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
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UniProtKB/SwissProt
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In DepthDetails
Affinity DataKd: 13nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataKd: 229nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataKd: 12nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
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UniProtKB/SwissProt
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In DepthDetails
Affinity DataKd: 600nMAssay Description:Tested for its antagonist activity against (DPDE)delta receptor in mouse vas deferensMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
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In DepthDetails