Compile Data Set for Download or QSAR
Found 9 Enz. Inhib. hit(s) with all data for entry = 50018207
LigandPNGBDBM50406141(CHEMBL5286547)copy SMILEScopy InChI
Affinity DataKi:  1.80E+3nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50406139(CHEMBL5281816)copy SMILEScopy InChI
Affinity DataKi:  3.60E+3nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50406140(CHEMBL5284779)copy SMILEScopy InChI
Affinity DataKi:  4.00E+3nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50406144(CHEMBL5283506)copy SMILEScopy InChI
Affinity DataKi:  1.10E+4nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50406145(CHEMBL5287800)copy SMILEScopy InChI
Affinity DataKi:  1.70E+4nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50406143(CHEMBL5287916)copy SMILEScopy InChI
Affinity DataKi:  1.90E+4nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50406142(CHEMBL5280788)copy SMILEScopy InChI
Affinity DataKi:  3.70E+4nMAssay Description:Antagonistic activity against M2 muscarinic receptor in guinea pig left atrium derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails
TargetNuclear receptor ROR-alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50406142(CHEMBL5280788)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+4nMAssay Description:In vitro antagonism of OT-induced uterine contractions,against rat uterus by measuring pA2 value which refers to the negative logarithm of the molar ...More data for this Ligand-Target Pair
In DepthDetails
TargetNuclear receptor ROR-beta(Homo sapiens (Human))TBA
LigandPNGBDBM50406142(CHEMBL5280788)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+4nMAssay Description:Antagonist activity against CCK-8 induced responses in guinea pig gall bladder was determinedMore data for this Ligand-Target Pair
In DepthDetails