Affinity DataKi: 15nMAssay Description:Relative potency against Histamine H1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataKi: 120nMAssay Description:Apparent pA2 value of compound at 50 nM concentration of mepyramine in rat aortaMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataKi: 2.41E+3nMAssay Description:Apparent pA2 value of compound at 10 nM concentration of mepyramine in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataKi: 3.12E+3nMAssay Description:Antagonistic activity for carbachol induced contractions in guinea pig ileum against Muscarinic acetylcholine receptor M3 in the presence of mepyrami...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataKi: 3.80E+3nMAssay Description:Antagonistic activity for carbachol induced contractions in guinea pig ileum against Muscarinic acetylcholine receptor M3 in the presence of mepyrami...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataKi: 4.46E+4nMAssay Description:Tetsed for Antagonistic activity at histamine H3 receptor in guinea pig ileal longitudinal muscle in the presence of mepyramine at a concentration of...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 0.100nMAssay Description:Antagonistic activity for carbachol induced contractions in guinea pig ileum against Muscarinic acetylcholine receptor M3 in the presence of mepyrami...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 3nMAssay Description:Antagonistic affinity tested against isolated Rat Thoracic Aorta Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 4nMAssay Description:Tetsed for Antagonistic activity at histamine H3 receptor in guinea pig ileal longitudinal muscle in the presence of mepyramine at a concentration of...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 5nMAssay Description:Tetsed for Antagonistic activity at histamine H3 receptor in guinea pig ileal longitudinal muscle in the presence of mepyramine at a concentration of...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 9.40nMAssay Description:Antagonistic affinity tested against isolated Rat Thoracic Aorta Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 11nMAssay Description:Tetsed for Antagonistic activity at histamine H3 receptor in guinea pig ileal longitudinal muscle in the presence of mepyramine at a concentration of...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 25nMAssay Description:Apparent pA2 value of compound at 10 nM concentration of mepyramine in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 30nMAssay Description:Tetsed for Antagonistic activity at histamine H3 receptor in guinea pig ileal longitudinal muscle in the presence of mepyramine at a concentration of...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 46nMAssay Description:Antagonistic activity for carbachol induced contractions in guinea pig ileum against Muscarinic acetylcholine receptor M3 in the presence of mepyrami...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 49nMAssay Description:Histamine-induced inhibition of forskolin- stimulated cAMP accumulation in SK-N-MC cells overexpressing the human Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 97nMAssay Description:Antagonistic affinity tested against isolated Rat Thoracic Aorta Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 188nMAssay Description:In vitro relative antagonist potency towards guinea pig Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 303nMAssay Description:Antagonistic affinity tested against isolated Rat Prostatic Vas Deferens Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 570nMAssay Description:Antagonistic activity for carbachol induced contractions in guinea pig ileum against Muscarinic acetylcholine receptor M3 in the presence of mepyrami...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 850nMAssay Description:Maximum response (E max) against Histamine H1 receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro relative antagonist potency towards guinea pig Tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 1.07E+3nMAssay Description:Histamine-induced inhibition of forskolin- stimulated cAMP accumulation in SK-N-MC cells overexpressing the human Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 1.09E+3nMAssay Description:Apparent pA2 value of compound at 50 nM concentration of mepyramine in rat aortaMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 1.39E+3nMAssay Description:Histamine-induced inhibition of forskolin- stimulated cAMP accumulation in SK-N-MC cells overexpressing the human Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 1.90E+3nMAssay Description:Apparent pA2 value of compound at 10 nM concentration of mepyramine in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 2.04E+3nMAssay Description:Histamine-induced inhibition of forskolin- stimulated cAMP accumulation in SK-N-MC cells overexpressing the human Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 6.58E+3nMAssay Description:Antagonistic activity for carbachol induced contractions in guinea pig ileum against Muscarinic acetylcholine receptor M3 in the presence of mepyrami...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 7.97E+3nMAssay Description:Tetsed for Antagonistic activity at histamine H3 receptor in guinea pig ileal longitudinal muscle in the presence of mepyramine at a concentration of...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 1.01E+4nMAssay Description:Antagonistic activity for carbachol induced contractions in guinea pig ileum against Muscarinic acetylcholine receptor M3 in the presence of mepyrami...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 1.22E+4nMAssay Description:Relative potency against Histamine H1 receptor in endothelium-Denuded rings of guinea pig AortaMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 5.00E+4nMAssay Description:Apparent pA2 value of compound at 10 nM concentration of mepyramine in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 5.00E+4nMAssay Description:Histamine-induced inhibition of forskolin- stimulated cAMP accumulation in SK-N-MC cells overexpressing the human Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 5.00E+4nMAssay Description:Histamine-induced inhibition of forskolin- stimulated cAMP accumulation in SK-N-MC cells overexpressing the human Histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 5.00E+4nMAssay Description:Tetsed for Antagonistic activity at histamine H3 receptor in guinea pig ileal longitudinal muscle in the presence of mepyramine at a concentration of...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 5.00E+4nMAssay Description:Apparent pA2 value of compound at 50 nM concentration of mepyramine in rat aortaMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 5.00E+4nMAssay Description:Tetsed for Antagonistic activity at histamine H3 receptor in guinea pig ileal longitudinal muscle in the presence of mepyramine at a concentration of...More data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 1.35E+5nMAssay Description:Antagonistic activity for carbachol induced contractions in guinea pig ileum against Muscarinic acetylcholine receptor M3 in the presence of mepyrami...More data for this Ligand-Target Pair
In DepthDetails
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