TargetEstrogen receptor beta(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Binding affinity to human ER betaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Binding affinity to human ER alphaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Binding affinity to ERalpha L384M/M421G mutantMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Binding affinity to ERalpha L384M/M421G mutantMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Binding affinity to ERalpha L384M/M421G mutantMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Binding affinity to ERalpha L384M/M421G mutantMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Binding affinity to ERalpha L384M/M421G mutantMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Binding affinity to ERalpha L384M/M421G mutantMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Binding affinity to ERalpha L384M/M421G mutantMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Binding affinity to ERalpha L384M/M421G mutantMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Binding affinity to ERalpha L384M/M421G mutantMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 82nMAssay Description:Binding affinity to ERalpha L384M/M421G mutantMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Binding affinity to human ER betaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Binding affinity to ERalpha L384M/M421G mutantMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Binding affinity to human ER betaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Binding affinity to ERalpha L384M/M421G mutantMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Binding affinity to ERalpha L384M/M421G mutantMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Binding affinity to human ER betaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Binding affinity to human ER alphaMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Binding affinity to human ER betaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Binding affinity to human ER alphaMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 310nMAssay Description:Binding affinity to human ER betaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Binding affinity to ERalpha L384M/M421G mutantMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Binding affinity to human ER alphaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Binding affinity to ERalpha L384M/M421G mutantMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 510nMAssay Description:Binding affinity to human ER betaMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Binding affinity to human ER betaMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Binding affinity to human ER betaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 620nMAssay Description:Binding affinity to human ER alphaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 710nMAssay Description:Binding affinity to human ER alphaMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity to human ER betaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Binding affinity to human ER alphaMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Binding affinity to human ER betaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Binding affinity to human ER alphaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Binding affinity to ERalpha L384M/M421G mutantMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Binding affinity to human ER alphaMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Binding affinity to human ER betaMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Binding affinity to human ER betaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Binding affinity to wild type ERalphaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:Binding affinity to human ER alphaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 3.90E+3nMAssay Description:Binding affinity to ERalpha L384M/M421G mutantMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 5.50E+3nMAssay Description:Binding affinity to ERalpha L384M/M421G mutantMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:Binding affinity to human ER betaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 6.80E+3nMAssay Description:Binding affinity to wild type ERalphaMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to human ER betaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to human ER alphaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to human ER alphaMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to human ER betaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to human ER alphaMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
IRBM (Merck Research Laboratories Rome)
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to human ER alphaMore data for this Ligand-Target Pair