Compile Data Set for Download or QSAR
Found 97 Enz. Inhib. hit(s) with all data for entry = 50018309
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421673(CHEMBL5283441)copy SMILEScopy InChI
Affinity DataKi:  290nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421686(CHEMBL5282194)copy SMILEScopy InChI
Affinity DataKi:  320nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50293150(CHEMBL468963 | D3RKN_26 | GSK screening, 38 | N-(4...)copy SMILEScopy InChI
Affinity DataKi:  420nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421679(CHEMBL5282708)copy SMILEScopy InChI
Affinity DataKi:  440nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421671(CHEMBL5266831)copy SMILEScopy InChI
Affinity DataKi:  470nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421672(CHEMBL5316225)copy SMILEScopy InChI
Affinity DataKi:  580nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421685(CHEMBL5280226)copy SMILEScopy InChI
Affinity DataKi:  700nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421687(CHEMBL5277580)copy SMILEScopy InChI
Affinity DataKi:  970nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421681(CHEMBL5273566)copy SMILEScopy InChI
Affinity DataKi:  1.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421683(CHEMBL5283041)copy SMILEScopy InChI
Affinity DataKi:  1.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421676(CHEMBL5283475)copy SMILEScopy InChI
Affinity DataKi:  1.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421680(CHEMBL5277737)copy SMILEScopy InChI
Affinity DataKi:  1.50E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421682(CHEMBL5285809)copy SMILEScopy InChI
Affinity DataKi:  1.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421684(CHEMBL5277619)copy SMILEScopy InChI
Affinity DataKi:  1.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421674(CHEMBL5284844)copy SMILEScopy InChI
Affinity DataKi:  2.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421678(CHEMBL5286085)copy SMILEScopy InChI
Affinity DataKi:  2.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421675(CHEMBL5266857)copy SMILEScopy InChI
Affinity DataKi:  2.70E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421677(CHEMBL5280561)copy SMILEScopy InChI
Affinity DataKi: >1.20E+4nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50421681(CHEMBL5273566)copy SMILEScopy InChI
Affinity DataIC50: 180nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421673(CHEMBL5283441)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421686(CHEMBL5282194)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50293150(CHEMBL468963 | D3RKN_26 | GSK screening, 38 | N-(4...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50293150(CHEMBL468963 | D3RKN_26 | GSK screening, 38 | N-(4...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421679(CHEMBL5282708)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421671(CHEMBL5266831)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421672(CHEMBL5316225)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421685(CHEMBL5280226)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421687(CHEMBL5277580)copy SMILEScopy InChI
Affinity DataIC50: 3.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421681(CHEMBL5273566)copy SMILEScopy InChI
Affinity DataIC50: 3.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421683(CHEMBL5283041)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421676(CHEMBL5283475)copy SMILEScopy InChI
Affinity DataIC50: 4.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50421672(CHEMBL5316225)copy SMILEScopy InChI
Affinity DataIC50: 4.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421680(CHEMBL5277737)copy SMILEScopy InChI
Affinity DataIC50: 5.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421682(CHEMBL5285809)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421684(CHEMBL5277619)copy SMILEScopy InChI
Affinity DataIC50: 6.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50421673(CHEMBL5283441)copy SMILEScopy InChI
Affinity DataIC50: 7.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50421674(CHEMBL5284844)copy SMILEScopy InChI
Affinity DataIC50: 7.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421674(CHEMBL5284844)copy SMILEScopy InChI
Affinity DataIC50: 7.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421678(CHEMBL5286085)copy SMILEScopy InChI
Affinity DataIC50: 8.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50421671(CHEMBL5266831)copy SMILEScopy InChI
Affinity DataIC50: 9.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)TBA
LigandPNGBDBM50421675(CHEMBL5266857)copy SMILEScopy InChI
Affinity DataIC50: 9.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50421684(CHEMBL5277619)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50421677(CHEMBL5280561)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+4nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50421680(CHEMBL5277737)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50421682(CHEMBL5285809)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+4nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50421675(CHEMBL5266857)copy SMILEScopy InChI
Affinity DataIC50: 3.90E+4nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50421686(CHEMBL5282194)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50421685(CHEMBL5280226)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50421683(CHEMBL5283041)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50421679(CHEMBL5282708)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
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