Affinity DataKi: 0.840nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.47nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute for Degenerative Diseases
Curated by ChEMBL
Institute for Degenerative Diseases
Curated by ChEMBL
Affinity DataKi: 14.2nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 15.4nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 27.6nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 28.5nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Institute for Degenerative Diseases
Curated by ChEMBL
Institute for Degenerative Diseases
Curated by ChEMBL
Affinity DataKi: 40.4nMAssay Description:Displacement of [3H]paroxetine from SERT in brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 70.4nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 71.9nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 73.8nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 79.6nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 101nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Institute for Degenerative Diseases
Curated by ChEMBL
Institute for Degenerative Diseases
Curated by ChEMBL
Affinity DataKi: 141nMAssay Description:Displacement of [3H]paroxetine from SERT in brain membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute for Degenerative Diseases
Curated by ChEMBL
Institute for Degenerative Diseases
Curated by ChEMBL
Affinity DataKi: 186nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute for Degenerative Diseases
Curated by ChEMBL
Institute for Degenerative Diseases
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute for Degenerative Diseases
Curated by ChEMBL
Institute for Degenerative Diseases
Curated by ChEMBL
Affinity DataKi: 228nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Institute for Degenerative Diseases
Curated by ChEMBL
Institute for Degenerative Diseases
Curated by ChEMBL
Affinity DataKi: 252nMAssay Description:Displacement of [3H]paroxetine from SERT in brain membranesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Institute for Degenerative Diseases
Curated by ChEMBL
Institute for Degenerative Diseases
Curated by ChEMBL
Affinity DataKi: 351nMAssay Description:Displacement of [3H]paroxetine from SERT in brain membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute for Degenerative Diseases
Curated by ChEMBL
Institute for Degenerative Diseases
Curated by ChEMBL
Affinity DataKi: 410nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Institute for Degenerative Diseases
Curated by ChEMBL
Institute for Degenerative Diseases
Curated by ChEMBL
Affinity DataKi: 486nMAssay Description:Displacement of [3H]paroxetine from SERT in brain membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute for Degenerative Diseases
Curated by ChEMBL
Institute for Degenerative Diseases
Curated by ChEMBL
Affinity DataKi: 716nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute for Degenerative Diseases
Curated by ChEMBL
Institute for Degenerative Diseases
Curated by ChEMBL
Affinity DataKi: 740nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute for Degenerative Diseases
Curated by ChEMBL
Institute for Degenerative Diseases
Curated by ChEMBL
Affinity DataKi: 1.87E+3nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute for Degenerative Diseases
Curated by ChEMBL
Institute for Degenerative Diseases
Curated by ChEMBL
Affinity DataKi: 3.14E+3nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute for Degenerative Diseases
Curated by ChEMBL
Institute for Degenerative Diseases
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair