Compile Data Set for Download or QSAR
Found 11 Enz. Inhib. hit(s) with all data for entry = 50019151
TargetActivated CDC42 kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
In DepthDetails
TargetActivated CDC42 kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM4552(4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-...)copy SMILEScopy InChI
Affinity DataIC50: 2.70nMMore data for this Ligand-Target Pair
In DepthDetails
TargetActivated CDC42 kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50396483(PLX-4032 | RG 7204 | Ro 5185426 | US10570155, Vemu...)copy SMILEScopy InChI
Affinity DataIC50: 19nMMore data for this Ligand-Target Pair
In DepthDetails
TargetActivated CDC42 kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50436850(CERITINIB | CHEMBL2403108 | LDK378 | US10053458, C...)copy SMILEScopy InChI
Affinity DataIC50: 34nMMore data for this Ligand-Target Pair
In DepthDetails
TargetActivated CDC42 kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50029668(AZD-9291 | Osimertinib | US10085983, Compound AZD-...)copy SMILEScopy InChI
Affinity DataIC50: 71nMMore data for this Ligand-Target Pair
In DepthDetails
TargetActivated CDC42 kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM3603(4-N-(3-bromophenyl)-6-N-methylpyrido[3,4-d]pyrimid...)copy SMILEScopy InChI
Affinity DataIC50: 200nMMore data for this Ligand-Target Pair
In DepthDetails
TargetActivated CDC42 kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)copy SMILEScopy InChI
Affinity DataIC50: 7.83E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetActivated CDC42 kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
TargetActivated CDC42 kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
TargetActivated CDC42 kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataKd:  5.60nMMore data for this Ligand-Target Pair
In DepthDetails
TargetActivated CDC42 kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50337126(2-(2-methoxy-4-(4-methylpiperazin-1-yl)phenylamino...)copy SMILEScopy InChI
Affinity DataKd:  15nMMore data for this Ligand-Target Pair
In DepthDetails