Compile Data Set for Download or QSAR
Found 42 Enz. Inhib. hit(s) with all data for entry = 50020285
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212166(7-chloro-6H-chromeno[4,3-b]quinoline-3,9-diol | CH...)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212173(7-bromo-6H-chromeno[4,3-b]quinoline-3,9-diol | CHE...)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171724(4-Bromo-2-(4-hydroxy-phenyl)-quinolin-6-ol | 4-bro...)copy SMILEScopy InChI
Affinity DataIC50: 4.30nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171726(4-Chloro-2-(4-hydroxy-phenyl)-quinolin-6-ol | 4-ch...)copy SMILEScopy InChI
Affinity DataIC50: 4.60nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212172(3,9-dihydroxy-6H-chromeno[4,3-b]quinoline-7-carbon...)copy SMILEScopy InChI
Affinity DataIC50: 6.10nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212161(7-vinyl-6H-chromeno[4,3-b]quinoline-3,9-diol | CHE...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171712(6-Hydroxy-2-(4-hydroxy-phenyl)-quinoline-4-carboni...)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212162(7-ethyl-6H-chromeno[4,3-b]quinoline-3,9-diol | CHE...)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171723(4-Ethyl-2-(4-hydroxy-phenyl)-quinolin-6-ol | 4-eth...)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212170(7-ethynyl-6H-chromeno[4,3-b]quinoline-3,9-diol | C...)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212173(7-bromo-6H-chromeno[4,3-b]quinoline-3,9-diol | CHE...)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171727(2-(4-Hydroxy-phenyl)-4-vinyl-quinolin-6-ol | 2-(4-...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212168(4-(3,9-dihydroxy-6H-chromeno[4,3-b]quinolin-7-yl)b...)copy SMILEScopy InChI
Affinity DataIC50: 65nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171729(4-Ethynyl-2-(4-hydroxy-phenyl)-quinolin-6-ol | 4-e...)copy SMILEScopy InChI
Affinity DataIC50: 75nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212167(7-(3-methoxyphenyl)-6H-chromeno[4,3-b]quinoline-3,...)copy SMILEScopy InChI
Affinity DataIC50: 86nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212166(7-chloro-6H-chromeno[4,3-b]quinoline-3,9-diol | CH...)copy SMILEScopy InChI
Affinity DataIC50: 88nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212163(7-(4-methoxyphenyl)-6H-chromeno[4,3-b]quinoline-3,...)copy SMILEScopy InChI
Affinity DataIC50: 94nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212172(3,9-dihydroxy-6H-chromeno[4,3-b]quinoline-7-carbon...)copy SMILEScopy InChI
Affinity DataIC50: 98nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212165(7-(3-chlorophenyl)-6H-chromeno[4,3-b]quinoline-3,9...)copy SMILEScopy InChI
Affinity DataIC50: 144nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212169(3-(3,9-dihydroxy-6H-chromeno[4,3-b]quinolin-7-yl)b...)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212164(7-(4-chlorophenyl)-6H-chromeno[4,3-b]quinoline-3,9...)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171724(4-Bromo-2-(4-hydroxy-phenyl)-quinolin-6-ol | 4-bro...)copy SMILEScopy InChI
Affinity DataIC50: 212nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171726(4-Chloro-2-(4-hydroxy-phenyl)-quinolin-6-ol | 4-ch...)copy SMILEScopy InChI
Affinity DataIC50: 213nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212171(7-(4-(trifluoromethyl)phenyl)-6H-chromeno[4,3-b]qu...)copy SMILEScopy InChI
Affinity DataIC50: 319nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)copy SMILEScopy InChI
Affinity DataIC50: 395nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171712(6-Hydroxy-2-(4-hydroxy-phenyl)-quinoline-4-carboni...)copy SMILEScopy InChI
Affinity DataIC50: 455nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212165(7-(3-chlorophenyl)-6H-chromeno[4,3-b]quinoline-3,9...)copy SMILEScopy InChI
Affinity DataIC50: 504nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171727(2-(4-Hydroxy-phenyl)-4-vinyl-quinolin-6-ol | 2-(4-...)copy SMILEScopy InChI
Affinity DataIC50: 504nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212161(7-vinyl-6H-chromeno[4,3-b]quinoline-3,9-diol | CHE...)copy SMILEScopy InChI
Affinity DataIC50: 526nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212163(7-(4-methoxyphenyl)-6H-chromeno[4,3-b]quinoline-3,...)copy SMILEScopy InChI
Affinity DataIC50: 549nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212170(7-ethynyl-6H-chromeno[4,3-b]quinoline-3,9-diol | C...)copy SMILEScopy InChI
Affinity DataIC50: 624nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171723(4-Ethyl-2-(4-hydroxy-phenyl)-quinolin-6-ol | 4-eth...)copy SMILEScopy InChI
Affinity DataIC50: 634nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212162(7-ethyl-6H-chromeno[4,3-b]quinoline-3,9-diol | CHE...)copy SMILEScopy InChI
Affinity DataIC50: 641nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212167(7-(3-methoxyphenyl)-6H-chromeno[4,3-b]quinoline-3,...)copy SMILEScopy InChI
Affinity DataIC50: 820nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212168(4-(3,9-dihydroxy-6H-chromeno[4,3-b]quinolin-7-yl)b...)copy SMILEScopy InChI
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212169(3-(3,9-dihydroxy-6H-chromeno[4,3-b]quinolin-7-yl)b...)copy SMILEScopy InChI
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171729(4-Ethynyl-2-(4-hydroxy-phenyl)-quinolin-6-ol | 4-e...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212164(7-(4-chlorophenyl)-6H-chromeno[4,3-b]quinoline-3,9...)copy SMILEScopy InChI
Affinity DataIC50: 2.35E+3nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212171(7-(4-(trifluoromethyl)phenyl)-6H-chromeno[4,3-b]qu...)copy SMILEScopy InChI
Affinity DataIC50: 5.24E+3nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V124HVPubMed