TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 0.520nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 0.720nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 3.70nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 6.70nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 8.20nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 52nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 54nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 54nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 76nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 79nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 81nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 83nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 86nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 132nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 136nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 137nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 144nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 174nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 177nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 212nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 343nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 627nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 670nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 755nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 790nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 810nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 870nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 907nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 1.02E+3nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair