TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataKi: 72nMAssay Description:Binding affinity at GPR109aMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataKi: 156nMAssay Description:Binding affinity at GPR109aMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataKi: 3.50E+3nMAssay Description:Binding affinity at GPR109aMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Activity at GPR109a (unknown origin) assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Activity at GPR109a (unknown origin) assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 3(Homo sapiens (Human))
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Activity at GPR109b assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataEC50: 200nMAssay Description:Activity at GPR109a (unknown origin) assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataEC50: 400nMAssay Description:Activity at GPR109a (unknown origin) assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 3(Homo sapiens (Human))
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataEC50: 1.72E+3nMAssay Description:Activity at GPR109b assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 3(Homo sapiens (Human))
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataEC50: 1.47E+3nMAssay Description:Activity at GPR109b assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataEC50: 110nMAssay Description:Activity at GPR109a (unknown origin) assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair